Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2006-06-08
2009-02-17
Rao, Deepak (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C514S277000, C514S235800, C544S058600, C544S122000, C544S323000
Reexamination Certificate
active
07491732
ABSTRACT:
The invention encompasses compounds having formula I-V and the compositions and methods using these compounds in the treatment of conditions in which modulation of the JAK pathway or inhibition of JAK kinases, particularly JAK3, may be therapeutically useful.
REFERENCES:
patent: 4166452 (1979-09-01), Generales, Jr.
patent: 4256108 (1981-03-01), Theeuwes
patent: 4265874 (1981-05-01), Bonsen et al.
patent: 5700904 (1997-12-01), Baker et al.
patent: 5728536 (1998-03-01), Ihle et al.
patent: 6080747 (2000-06-01), Uckun et al.
patent: 6080748 (2000-06-01), Uckun et al.
patent: 6133305 (2000-10-01), Tang et al.
patent: 6177433 (2001-01-01), Uckun et al.
patent: 6210654 (2001-04-01), Ihle et al.
patent: 6313130 (2001-11-01), Uckun et al.
patent: 6316635 (2001-11-01), Tang et al.
patent: 6433018 (2002-08-01), Siddiqui et al.
patent: 6486185 (2002-11-01), McMahon et al.
patent: 6506763 (2003-01-01), Tang et al.
patent: 6528509 (2003-03-01), Hale et al.
patent: 6593357 (2003-07-01), Green et al.
patent: 6608048 (2003-08-01), Tsou et al.
patent: 6610688 (2003-08-01), Liang et al.
patent: 6635651 (2003-10-01), Uckun
patent: 6677368 (2004-01-01), Cui et al.
patent: 6683082 (2004-01-01), Tang et al.
patent: 6696448 (2004-02-01), Tang et al.
patent: 6699865 (2004-03-01), Hale et al.
patent: 6710052 (2004-03-01), Pease et al.
patent: 6777417 (2004-08-01), Liang et al.
patent: 6784195 (2004-08-01), Hale et al.
patent: 6815439 (2004-11-01), Harris et al.
patent: 6825190 (2004-11-01), Moon et al.
patent: 6908920 (2005-06-01), Thomas et al.
patent: 6949580 (2005-09-01), Hale et al.
patent: 6969760 (2005-11-01), Ihle et al.
patent: 6998391 (2006-02-01), Lyons et al.
patent: 7056944 (2006-06-01), Hale et al.
patent: 7074793 (2006-07-01), Hudkins et al.
patent: 7105529 (2006-09-01), Davis et al.
patent: 2001/0007033 (2001-07-01), Tang et al.
patent: 2002/0115173 (2002-08-01), Ben-Sasson
patent: 2002/0137141 (2002-09-01), Ben-Sasson
patent: 2003/0149064 (2003-08-01), Pease et al.
patent: 2003/0236244 (2003-12-01), Ledford
patent: 2004/0029902 (2004-02-01), Singh et al.
patent: 2004/0102455 (2004-05-01), Burns et al.
patent: 2004/0142404 (2004-07-01), Wilks et al.
patent: 2004/0147507 (2004-07-01), Ledeboer et al.
patent: 2004/0214817 (2004-10-01), Pierce et al.
patent: 2005/0176743 (2005-08-01), Luecking et al.
patent: 2005/0209224 (2005-09-01), Singh
patent: 2005/0234049 (2005-10-01), Singh et al.
patent: 2006/0167254 (2006-07-01), Cooper et al.
patent: 2006/0211657 (2006-09-01), Singh et al.
patent: 2006/0270694 (2006-11-01), Wong
patent: 2007/0203161 (2007-08-01), Argade
patent: 02463989 (2004-04-01), None
patent: 2542492 (2005-04-01), None
patent: WO 95/03701 (1995-02-01), None
patent: WO 99/15500 (1999-04-01), None
patent: WO 00/00202 (2000-01-01), None
patent: WO 00/10981 (2000-03-01), None
patent: WO 00/27825 (2000-05-01), None
patent: WO 00/39101 (2000-07-01), None
patent: WO 00/47583 (2000-08-01), None
patent: WO 00/51587 (2000-09-01), None
patent: WO 00/55159 (2000-09-01), None
patent: WO 00/78731 (2000-12-01), None
patent: WO 01/42246 (2001-06-01), None
patent: WO 01/45641 (2001-06-01), None
patent: WO 01/52892 (2001-07-01), None
patent: WO 01/56993 (2001-08-01), None
patent: WO 01/57022 (2001-08-01), None
patent: WO 01/64654 (2001-09-01), None
patent: WO 03/094920 (2001-09-01), None
patent: WO 01/72758 (2001-10-01), None
patent: WO 02/00661 (2002-01-01), None
patent: WO 02/04429 (2002-01-01), None
patent: WO 02/43735 (2002-06-01), None
patent: WO 02/48336 (2002-06-01), None
patent: WO 02/059110 (2002-08-01), None
patent: WO 02/060492 (2002-08-01), None
patent: WO 02/060927 (2002-08-01), None
patent: WO 02/096888 (2002-12-01), None
patent: WO 02/096909 (2002-12-01), None
patent: WO 02/102313 (2002-12-01), None
patent: WO 02/102800 (2002-12-01), None
patent: WO 03/000186 (2003-01-01), None
patent: WO 03/002542 (2003-01-01), None
patent: WO 03/018021 (2003-03-01), None
patent: WO 03/018022 (2003-03-01), None
patent: WO 03/020698 (2003-03-01), None
patent: WO 03/030909 (2003-04-01), None
patent: WO 03/032994 (2003-04-01), None
patent: WO 03/032997 (2003-04-01), None
patent: WO 03/048162 (2003-06-01), None
patent: WO 03/063794 (2003-08-01), None
patent: WO 03/066601 (2003-08-01), None
patent: WO 03/074515 (2003-09-01), None
patent: WO 03/078404 (2003-09-01), None
patent: WO 03/101989 (2003-12-01), None
patent: WO 03/106416 (2003-12-01), None
patent: WO 2004/014382 (2004-02-01), None
patent: WO 2004/016597 (2004-02-01), None
patent: WO 2004/041789 (2004-05-01), None
patent: WO 2004/041810 (2004-05-01), None
patent: WO 2004/041814 (2004-05-01), None
patent: WO 2004/043467 (2004-05-01), None
patent: WO 2004/043953 (2004-05-01), None
patent: WO 2004/046112 (2004-06-01), None
patent: WO 2004/046118 (2004-06-01), None
patent: WO 2004/046120 (2004-06-01), None
patent: WO 2004/047843 (2004-06-01), None
patent: WO 2004/058749 (2004-07-01), None
patent: WO 2004/058753 (2004-07-01), None
patent: WO 2004/074244 (2004-09-01), None
patent: WO 2004/074261 (2004-09-01), None
patent: WO 2004/074262 (2004-09-01), None
patent: WO 2004/080980 (2004-09-01), None
patent: WO 2004/085388 (2004-10-01), None
patent: WO 2004/092154 (2004-10-01), None
patent: WO 2004/099159 (2004-11-01), None
patent: WO 2004/101549 (2004-11-01), None
patent: WO 2004/101564 (2004-11-01), None
patent: WO 2005/007621 (2005-01-01), None
patent: WO 2005/007646 (2005-01-01), None
patent: WO 2005/009957 (2005-02-01), None
patent: WO 2005/009980 (2005-02-01), None
patent: WO 2005/012262 (2005-02-01), None
patent: WO 2005/012294 (2005-02-01), None
patent: WO 2005/012304 (2005-02-01), None
patent: WO 2005/012307 (2005-02-01), None
patent: WO 2005/013996 (2005-02-01), None
patent: WO 2005/016344 (2005-02-01), None
patent: WO 2005/016893 (2005-02-01), None
patent: WO 2005/016894 (2005-02-01), None
patent: WO 2005/026130 (2005-03-01), None
patent: WO 2005/026158 (2005-03-01), None
patent: WO 2005/028467 (2005-03-01), None
patent: WO 2005/028475 (2005-03-01), None
patent: WO 2005/028479 (2005-03-01), None
patent: WO 2005/033107 (2005-04-01), None
patent: WO 2005/037800 (2005-04-01), None
patent: WO 2005/051366 (2005-06-01), None
patent: WO 2005/061458 (2005-07-01), None
patent: WO 2005/066156 (2005-07-01), None
patent: WO 2005/075468 (2005-08-01), None
patent: WO 2005/080393 (2005-09-01), None
patent: WO 2005/107760 (2005-11-01), None
patent: WO 2005/118544 (2005-12-01), None
patent: WO 2006/034872 (2006-04-01), None
patent: WO 2006/074057 (2006-07-01), None
patent: WO 2006/133426 (2006-12-01), None
patent: WO 2007/006926 (2007-01-01), None
patent: WO 2007/053452 (2007-05-01), None
patent: WO 2007/085540 (2007-08-01), None
patent: WO 2007/098507 (2007-08-01), None
Vippagunta et al., Cyrstalline Solids, Advanced Drug Delivery Reviews, 48, pp. 3-26, 2001.
West, Solid Solutions, Solid State Chemistry and its applications, pp. 358 & 365, 1988.
Ulrich, Chapter 4: Crystallization, Kirk-Othmer Encyclopedia of Chemical Technology, Aug. 2002.
Bundgaard, Design of Prodrugs: Introduction, p. 1, 1985.
Silverman, Prodrugs and Drug Delivery Systems, The Organic Chemistry of Drug Design and Drug Action, pp. 352-400, 1992.
Rajinder et al., CAPLUS Abstract 142:219300 (2005).
Singh et al., CAPLUS Abstract 140:199334 (2004).
Boloor et al., CAPLUS Abstract 137:140534 (2002).
Damasio, Alzheimer's Disease and Related Dementias, Cecil Textbook of Medicine, 20thEdition, vol. 2, pp. 1992-1996, 1996.
Layzer, Degenerative diseases of the Nervous System, Cecil Textbook of Medicine, 20thEdition, vol. 2, pp. 2050-2057, 1996.
Casanova et al., PubMed Abstract (Rev Neurol 28(9):909-15) May 1999.
Traxler, Protein Tyrosine Kinase inhibitors in cancer treatment, Exp. Opin. Ther. Patents, 7(6):571-588, 1997.
Simone, Oncology: Introduction, Cecil Textbook of Medicine, 20thEdition, vol. 1, pp. 1004-1010, 1996.
El-Kerdawy, M.M., et al., “2,4-Bis (Substituted)-5-Nitropyrimidines of Expected Diurectic Action.”Egypt. J. Chem.29(2):247-251 (1986).
Bungaard, H. et al. “A novel solution-stable, water-soluble prodrug type for drugs containing a hydroxyl or an NH-acidic g
Argade Ankush
Carroll David
Cooper Robin
Li Hui
Singh Rajinder
Foley & Lardner LLP
Rao Deepak
Rigel Pharmaceuticals Inc.
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