Chemistry: natural resins or derivatives; peptides or proteins; – Peptides of 3 to 100 amino acid residues – Somatostatin ; related peptides
Patent
1996-07-31
1998-06-23
Tsang, Cecilia J.
Chemistry: natural resins or derivatives; peptides or proteins;
Peptides of 3 to 100 amino acid residues
Somatostatin ; related peptides
530317, 530328, 514 9, 514 11, 514 15, 514 16, C07K 764, A61K 3804, A61K 3812
Patent
active
057706875
ABSTRACT:
Novel peptide analogs are disclosed. The novel peptides are conformationally constrained backbone cyclized somatostatin analogs. Methods for synthesizing the somatostatin analogs and for producing libraries of the somatostatin analogs are also disclosed. Furthermore, pharmaceutical compositions comprising somatostatin analogs, and methods of using such compositions in the treatment of endocrine disorders, neoplasms and metabolic disorders are also disclosed.
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Gellerman Gary
Gilon Chaim
Hornik Vered
Seri-Levy Alon
Gupta Anish
Peptor Limited
Tsang Cecilia J.
Yissim Research Development Co. of Hebrew University of Jerusale
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