Drug – bio-affecting and body treating compositions – Inorganic active ingredient containing – Hydrochloric acid
Reexamination Certificate
2004-01-21
2008-11-18
Richter, Johann (Department: 1621)
Drug, bio-affecting and body treating compositions
Inorganic active ingredient containing
Hydrochloric acid
C562S405000
Reexamination Certificate
active
07452555
ABSTRACT:
The present disclosure relates to novel cocrystals and novel methods for cocrystallization. In particular, the disclosure includes cocrystals comprising a salt of an active agent, such as a chloride salt of an active pharmaceutical ingredient. The present disclosure also relates to methods of preparing cocrystals and methods for screening for solid state phases.
REFERENCES:
patent: 2665277 (1954-01-01), Homeyer et al.
patent: 5080832 (1992-01-01), Etter et al.
Gavezzotti Acc. Chem. Res. 1994, 27, 309-314.
International Search Report and Written Opinion, dated Jul. 18, 2005, from International Application No. PCT/US04/01699.
Aakeroy, C. B.Acta Crystallogr. Sect. B-Struct. Sci.1997, 53, 569-586.
Aakeroy, C. B.; Evans, T. A.; Seddon, K. R.; Palinko, I.New J. Chem.1999, 23, 145-152.
Aullon, G.; Bellamy, D.; Brammer, L.; Bruton, E. A.; Orpen, A. G.Chem. Commun.1998, 653-654.
Bartoszak-Adamska, E.; Wojciechowski, G.; Jaskolski, M.; Brzezinski, M.;Journal of Molecular Structure595 (2001) 21-28.
Bettinetti, G.; Caira, M. R.; Callegari, A.; Merli, M.; Sorrenti, M.; Tadini, C.J. Pharm. Sci.2000, 89, 478-489.
Bettis, J. W.; Lach, J. L.; Hood, J.American Journal of Hospital Pharmacy1973, 30, 240-243.
Bilton, C.; Allen, F. H.; Shields, G. P.; Howard, J. A. K.Acta Crystallogr. Sect. B-Struct. Sci.2000, 56, 849-856.
Braga, D.; Cojazzi, G.; Abati, A.; Maini, L.; Polito, M.; Scaccianoce, L.; Grepioni, F.J. Chem. Soc.-Dalton Trans.2000, 3969-3975.
Braga, D; Draper S.M.; Champeil, E.; Grepioni, F.;Journal of Organometallic Chemistry573 (1999) 73-77.
Braga, D.; Maini, L.; Polito, M.; Grepioni, F.Chem. Commun.2002, 2302-2303.
Cheung, E.Y. et al.,J. Am. Chem. Soc., 2003, 125, 14658-59.
Cheung, E., et al.; “Direct Structure Determination of a Multicomponent Molecular Crystal Prepared by a Solid-State Grinding Procedure,”J. Am. Chem. Soc.XXXX,XXX (2003).
Coe, S.; Kane, J. J.; Nguyen, T. L.; Toledo, L. M.; Wininger, E.; Fowler, F. W.; Lauher, J. W.J. Am. Chem. Soc.1997, 119, 86-93.
Dalhus, B.; Gorbitz, C. H.Acta Crystallogr. Sect. C-Cryst. Struct. Commun.1999, 55, 1547-1555.
Datta, S.; Grant, D.J.W.;Nature, Jan. 2004, vol. 3, 42-57.
Dega-Szafran, Z.; Katrusiak, A.; Szafran, M.J. Mol. Struct.2001, 570, 165-174.
Deng, J. et al.; Tetrahedron :Asymmetry11 (2000) 1729-1732.
Desiraju, G. R., The Royal Society of Chemistry 2003, 466-467.
Dunitz, J.D.;The Royal Society of Chemistry2003, 506.
Edwards, M. R.; Jones, W.; Motherwell, W. D. S.Cryst. Eng2002, 5, 25-36.
Fleischman, S. G.; Kuduva, S. S.; McMahon, J. A.; Moulton, B.; Walsh, R. D. B.; Rodriguez-Hornedo, N.; Zaworotko, M. J.Cryst. Growth Des.2003, 3, 909-919.
Goldberg, I.;J. Am. Chem. Soc.1982, 104, 7077-7084.
Gorbitz, C. H.; Hersleth, H. P.Acta Crystallogr. Sect. B-Struct. Sci.2000, 56, 526-534.
Gorbitz, C. H.Acta Crystallogr. Sect. C-Cryst. Struct. Commun.2000, 56, 500-502.
Hu, Z-Q et al.,Acta Cryst.(2002) C58, o612-o614.
Hubschle, C.B. , et al.,Acta Cryst., (2002) C58, o540-o542.
Iimura, N.; Ohashi, Y.; Hirata, H.Bull. Chem. Soc. Jpn.2000, 73, 1097-1103.
Karlsson, R.;Acta Cryst., (1972) B28, 2358.
Kumar, V. S. S.; Nangia, A.; Katz, A. K.; Carrell, H. L.Cryst. Growth Des.2002, 2, 313-318.
Kuroda, R.; Imai, Y.; Tajima, N.Chem. Commun.2002, 2848-2849.
Morgan, T.K. et al. ; 1986 American Chemical Society, 1398-1405.
Nangia, A.; Desiraju, G. R.Acta Crystallogr. Sect. A1998, 54, 934-944.
O'Dowd, C.; Kennedy, J. D.; Thornton-Pett, M.J. Organomet. Chem.2002, 657, 20-39.
Orita, A.; Jiang, L. S.; Nakano, T.; Ma, N. C.; Otera, J.Chem. Commun.2002, 1362-1363.
Oswald, I. D. H.; Allan, D. R.; McGregor, P. A.; Motherwell, W. D. S.; Parsons, S.; Pulham, C. R.Acta Crystallogr. Sect. B-Struct. Sci. (2002)58, 1057-1066.
Pierpont, C. G.; Lang, S. A.Acta Crystallogr. Sect. C-Cryst. Struct. Commun.1986, 42, 1085-1087.
Rai, U. S.; George, S.Thermochim. Acta1994, 243, 17-25.
Reddy, L.S.; Nangia, A.; Lynch, V.M.;Crystal Growth&Design, “Phenyl-Perfluorophenyl Synthon Mediated Cocrystallization of Carboxylic Acids and Amides,” XXXX, vol. 0., No. 0, 1-6 2003.
Remenar, J.F. et al.;Organic Process Research&Development2003, 7, 990-996.
Remenar, J. F.; Morissette, S. L.; Peterson, M. L.; Moulton, B.; MacPhee, J. M.; Guzman, H. R.; Almarsson, O.J. Am. Chem. Soc.2003, 125, 8456-8457.
Rothenberg, G.; Downie, A. P.; Raston, C. L.; Scott, J. L.J. Am. Chem. Soc.2001, 123, 8701-8708.
Schauer, C.L. et al.,J. Chem. Soc., 1997, 119, 10245-10246.
Shan, N.; Toda, F.; Jones, W.Chem. Commun.2002, 2372-2373.
Steiner, T.Acta Crystallogr. Sect. B-Struct. Sci.1998, 54, 456-463.
Steiner, T.New J. Chem.1998, 22, 1099-1103.
Thallapally, P. K.; Nangia, A.Crystengcomm2001, art. No. 27.
TransForm Pharmaceuticals, Inc. Press Release, Lexington, MA, Nov. 3, 2003.
Videnova-Adrabinska, V.Acta Cryst.1996, B52, 1048-1056.
Vishweshwar, P.; Nangia, A.; Lynch, V. M.Cryst. Growth Des.2003, 3, 783-790.
Vishweshwar, P.; Nangia, A.; Lynch, V. M.Crystengcomm2003, 164-168.
Walsh, R. D. B.; Bradner, M. W.; Fleischman, S.; Morales, L. A.; Moulton, B.; Rodriguez-Hornedo, N.; Zaworotko, M. J.Chem. Commun.2003, 186-187.
Wang, K. W.; Pan, Y. J.; Jin, Z. M. Z.Krist.-New Cryst. Struct.2002, 217, 435-436.
Lindeman Jeffrey A.
Nixon & Peabody LLP
Richter Johann
S.S.C.I. Inc.
Valenrod Yevegeny
LandOfFree
Cocrystallization does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Cocrystallization, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Cocrystallization will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-4048458