Co-crystals and pharmaceutical compositions comprising the same

Details Co-crystals and pharmaceutical compositions comprising the same Co-crystals and pharmaceutical compositions comprising the same

2007-02-27

2011-10-18

Wilson, James O (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S255060

Reexamination Certificate

active

08039475

ABSTRACT:
The invention relates to compositions and co-crystals each comprising (1S,3aR,6aS)-2-[(2S)-2-[[(2S)-2-Cyclohexyl-2-(pyrazine-2-carbonylamino)acetyl]amino]-3,3-dimethylbutanoyl]-N-[(3S)-1-(cyclopropylamino)-1,2-dioxohexan-3-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrole-1-carboxamide having the structure:and the co-crystal former salicylic acid. Also within the scope of this invention are methods of making and using the same.

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