Cholesterol sequestrant glycosides that inhibit intestinal chole

Details Cholesterol sequestrant glycosides that inhibit intestinal chole Cholesterol sequestrant glycosides that inhibit intestinal chole

1993-06-21

1996-03-26

Robinson, Douglas W.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

514 53, 514 54, 536 5, 536 6, 5361231, 53612313, A61K 31705, A61K 31715, A01N 4500, A01N 4304

Patent

active

055020380

ABSTRACT:
Glycosides having neotigogenin aglycone moieties, administered orally to mammals are shown to inhibit the absorption of cholesterol. These compounds are useful in the treatment of hypercholesterolemia. Particular compounds are derived from tomato seeds and include neotigogenin trisaccharide.

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