Chemical synthesis of a highly potent epothilone

Details Chemical synthesis of a highly potent epothilone Chemical synthesis of a highly potent epothilone

2011-08-23

2011-08-23

Chandrakumar, Nizal (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C548S250000, C548S148000, C548S356100, C548S262200, C548S300100

Reexamination Certificate

active

08003801

ABSTRACT:
A highly active synthetic epothilone compound whose activity exceeds that of either epothilone EpoA or EpoB when assayed as a cytotoxic agent against a cancer cell line is disclosed as is a pharmaceutical composition containing the synthetic epothilone.

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