Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2007-02-20
2007-02-20
Berch, Mark L. (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C540S222000
Reexamination Certificate
active
10475845
ABSTRACT:
The present invention relates to a compound of the formula [I]: wherein A is lower alkylene or lower alkenylene; R1is lower alkyl, hydroxy(lower)alkyl, protected hydroxy(lower)alkyl, amino(lower)alkyl or protected amino(lower)alkyl, and R2is hydrogen or amino protecting group, or R1and R2are bonded together and form lower alkylene; R3and R5are independently amino or protected amino; and R4is carboxy or protected carboxy, or a pharmaceutically acceptable salt thereof, a process for preparing a compound of the formula [I], and a pharmaceutical composition comprising a compound of the formula [I] in admixture with a pharmaceutically acceptable carrier.
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Akamatsu Hisashi
Inoue Satoshi
Itoh Kenji
Kawabata Kohji
Misumi Keiji
Astellas Pharma Inc.
Berch Mark L.
Wakunaga Pharmaceutical Co., Ltd.
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