Cathepsin cysteine protease inhibitors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C514S252120, C514S252100, C514S256000, C514S311000, C514S357000, C514S381000, C514S399000, C514S521000, C544S170000, C544S335000, C544S392000, C546S152000, C546S330000, C558S410000

Reexamination Certificate

active

10525264

ABSTRACT:
This invention relates to class of compounds which are cysteine protease inhibitors, including but not limited to, inhibitors of cathepsins K, L, S and B. These compounds are useful for treating diseases in which inhibition of bone resorption is indicated, such as osteoporosis. They have the following structure: Formula (I)

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