Carvedilol

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Reexamination Certificate

active

07126008

ABSTRACT:
This invention relates to an improved process of preparing carvedilol, as well as a new crystalline hydrate and solvate and forms of carvedilol, processes for the manufacture thereof, and pharmaceutical compositions thereof.

REFERENCES:
patent: 4503067 (1985-03-01), Wiedemann et al.
patent: 5071868 (1991-12-01), Leinert
patent: 0 127 099 (1984-12-01), None
patent: 0 127 099 (1987-05-01), None
patent: 0 918 055 (1999-05-01), None
patent: WO 99/05105 (1999-02-01), None
G.M. Wall, “Pharmaceutical Applications of Drug Crystals Studies”, Pharmaceutical Manufacturing, vol. 3, No. 2, pp. 33-42, Feb. 1986.
J.K. Haleblian and W. McCrone, “Pharmaceutical Applications of Polymorphism”, Journal of Pharmaceutical Sciences, vol. 58, No. 8, pp. 911-929, Jul. 1969.
J.K. Haleblian, “Characterization of Habits and Crystalline Modifications of Solids and Their Pharmaceutical Applications”, Journal of Pharmaceutical Sciences, vol. 64, No. 8, pp. 1269-1288, Jul. 1975.
Pharmacopeial Forum, vol. 24, No. 1, pp. 5438-5441, Jan.-Feb. 1998.
Senderoff et al., “Synthesis of the Enantiomers and Three Racemic Metabolites of Carvedilol Labeled to High Specific Activity With Tritium”, Journal of Labeled Compounds and Radiopharmaceuticals, Dec. 1993, vol. 33, No. 12, pp. 1091-1105.
*Chen, Wei-Min et al. “Synthesis and Crystal Structure of Carvedilol” Jiegou Huaxue, vol. 17, No. 5, Sep. 1998, pp. 325-328 (abstract included).
*Carey, Francis A. et al. “Advanced Organic Chemistry” Third Edition, Part A: Structure and Mechanisms; Plenum Press, pp. 232-239. 1993.

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