Carboxylic acid derivative compounds and drugs comprising...

Details Carboxylic acid derivative compounds and drugs comprising... Carboxylic acid derivative compounds and drugs comprising...

2002-08-08

2009-02-17

Aulakh, Charanjit S (Department: 1625)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Radical -xh acid, or anhydride, acid halide or salt thereof...

C562S442000, C562S405000, C560S019000, C560S021000, C560S155000, C549S362000, C549S434000, C548S375100, C546S290000, C514S464000, C514S539000

Reexamination Certificate

active

07491748

ABSTRACT:
A carboxylic acid derivative of formula (I):wherein R1is —COOH, —COOR6, etc.; A is a single bond, alkylene, etc.; R2is alkyl, alkoxy, etc.; B is a carbocyclic ring or a heterocyclic ring; Q is alkylnene-Cyc2, etc.; D is a linking chain; and R3is alkyl, a carbocyclic ring or a heterocyclic ring, or a non-toxic salt thereof. The compound of formula (I) binds to PGE2receptor, especially subtypes EP3and/or EP4and show the antagonizing activity, are useful for the prevention and/or treatment of diseases induced pain, itch, urticaria, allergy, urinary frequency, urinary disturbance, Alzheimer's disease, cancer, dysmenorrhea, endometriosis, etc.

REFERENCES:
patent: 3950393 (1976-04-01), Keck et al.
patent: 4006246 (1977-02-01), Keck et al.
patent: RE29628 (1978-05-01), Keck et al.
patent: 4101671 (1978-07-01), Keck et al.
patent: 4113871 (1978-09-01), Stach et al.
patent: 4238506 (1980-12-01), Stach et al.
patent: 5268389 (1993-12-01), Harrison et al.
patent: 5412101 (1995-05-01), Caille et al.
patent: 5599830 (1997-02-01), Caille et al.
patent: 5684028 (1997-11-01), Caille et al.
patent: 5693827 (1997-12-01), Harrison et al.
patent: 5712298 (1998-01-01), Amschler
patent: 5716993 (1998-02-01), Ozaki et al.
patent: 5811445 (1998-09-01), Corbier et al.
patent: 5849796 (1998-12-01), Gericke et al.
patent: 5977155 (1999-11-01), Corbier et al.
patent: 6005116 (1999-12-01), Kojima et al.
patent: 6018068 (2000-01-01), Nagao et al.
patent: 6043275 (2000-03-01), Maruyama et al.
patent: 6462081 (2002-10-01), Maruyama et al.
patent: 0 073 663 (1983-03-01), None
patent: 0 081 993 (1983-06-01), None
patent: 985663 (2000-03-01), None
patent: 1 114 816 (2001-07-01), None
patent: WO 96/10569 (1996-04-01), None
patent: 97/05091 (1997-02-01), None
patent: WO 99/47497 (1999-09-01), None
patent: WO 00/03980 (2000-01-01), None
patent: WO 00/20371 (2000-01-01), None
patent: WO 00/15608 (2000-03-01), None
patent: WO 01/49661 (2001-07-01), None
patent: WO 02/16311 (2002-02-01), None
Russian Office Action dated Mar. 5, 2004.
International Search Report dated Dec. 17, 2002.

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