Organic compounds -- part of the class 532-570 series – Organic compounds – Carboxylic acids and salts thereof
Reexamination Certificate
2002-04-18
2009-06-09
Oh, Taylor Victor (Department: 1625)
Organic compounds -- part of the class 532-570 series
Organic compounds
Carboxylic acids and salts thereof
C562S405000, C562S488000
Reexamination Certificate
active
07544835
ABSTRACT:
Carboxylic acid compound or salt or hydrate thereof useful as insulin sensitizer, represented by the formulawherein R1represents hydrogen, hydroxyl, halogen, carboxyl, or C1-6alkyl, L represents single bond or C1-6-alkylene, C2-6-alkenylene, or C2-6-alkynylene, M represents single bond or C1-6-alkylene, C2-6-alkenylene, or C2-6-alkynylene, T represents single bond, or C1-3-alkylene, C2-3-alkenylene, or C2-3-alkynylene, W represents carboxyl,represents single bond, X represents single bond, oxygen, —NRX1CQ1O—, —OCQ1NRX1—, —CQ1NRX1O—, ONRX1CQ1—, —Q2SO2—, or —SO2Q2—, Y represents 5- to 14-membered aromatic group, and ring Z represents 5- to 14-membered aromatic group.
REFERENCES:
patent: 6506797 (2003-01-01), Nomura et al.
patent: 6884821 (2005-04-01), Shinoda et al.
patent: 7244861 (2007-07-01), Matsuura et al.
patent: 7253178 (2007-08-01), Matsuura et al.
patent: 2004/0102634 (2004-05-01), Matsuura et al.
patent: 2004/0116708 (2004-06-01), Harada et al.
patent: 2004/0138271 (2004-07-01), Matsuura et al.
patent: 2004/0214888 (2004-10-01), Matsuura et al.
patent: 2005/0014833 (2005-01-01), Clark et al.
patent: 3026924 (1982-02-01), None
patent: 0028063 (1981-05-01), None
patent: 0028063 (1984-06-01), None
patent: 219308 (1987-04-01), None
patent: 543662 (1993-05-01), None
patent: 1026149 (2000-08-01), None
patent: 57-64639 (1982-04-01), None
patent: 9-48771 (1997-02-01), None
patent: 11-152269 (1999-06-01), None
patent: 2001-55367 (2001-02-01), None
patent: 2001-261612 (2001-09-01), None
patent: WO 89/03819 (1989-05-01), None
patent: WO 90/06920 (1990-06-01), None
patent: WO 94/01420 (1994-01-01), None
patent: WO 94/13650 (1994-06-01), None
patent: WO 95/03288 (1995-02-01), None
patent: WO 99-04815 (1999-02-01), None
patent: WO 99/16758 (1999-04-01), None
patent: WO 99/18066 (1999-04-01), None
patent: WO-99/20275 (1999-04-01), None
patent: WO-99/36393 (1999-07-01), None
patent: WO-99/65897 (1999-12-01), None
patent: WO-00/04011 (2000-01-01), None
patent: WO 00/64876 (2000-11-01), None
patent: WO 00/64888 (2000-11-01), None
patent: WO 00/75103 (2000-12-01), None
patent: WO-01/21578 (2001-03-01), None
patent: WO-01/25181 (2001-04-01), None
patent: WO-01/25189 (2001-04-01), None
patent: WO-01/38325 (2001-05-01), None
patent: WO 01/55085 (2001-08-01), None
patent: WO 01/55086 (2001-08-01), None
patent: WO-01/92201 (2001-12-01), None
patent: WO-02/12210 (2002-02-01), None
patent: WO-02/34711 (2002-05-01), None
patent: WO-02/42273 (2002-05-01), None
patent: WO-02/079162 (2002-10-01), None
patent: WO-02/080899 (2002-10-01), None
patent: WO-02/081428 (2002-10-01), None
patent: WO-02/083616 (2002-10-01), None
patent: WO-02/100812 (2002-12-01), None
patent: WO-03/016265 (2003-02-01), None
patent: WO-03/055867 (2003-07-01), None
Paul W. Young et al., The Journal of Pharmacology and Experimental Therapeutics, 1997, vol. 284, No. 2, pp. 751 to 759.
David Haigh et al., Bioorganic & Medicinal Chemistry, 1999, vol. 7, No. 5, pp. 821 to 830.
“Nuovi Coloranti Per Miste Poliestere/Cotone” Tinctoria, 1996, vol. 93, No. 5, pp. 34 to 39.
D Gibson et al., European Journal of Medicinal Chemistry, 1997, vol. 32, No. 10, pp. 823 to 831.
Rico Lavoie et al., Bioorganic & Medicinal Chemistry Letters, 2001, vol. 11, No. 21, pp. 2847 to 2850.
Hulin et al., Current Pharmaceutical Design, 1996, 2, 85-102.
Buckle et al., Bioorganic & Medicinal Chemistry Letters, vol. 6, No. 17, pp. 2121-2126, 1996.
Bastie et al., The Journal of Biological Chemistry, vol. 274, No. 31, pp. 21920-21925, Jul. 30, 1999.
Lehmann et al., The Journal of Biological Chemistry, vol. 270, No. 22, 12953-12956, Jun. 2, 1995.
Willson et al., Journal of Medicinal Chemistry, vol. 43, No. 4, pp. 527-550 Feb. 24, 2000.
Barger et al., Trends in Cardiovasc. Med., vol. 10, No. 6, pp. 238-245, 2000.
Miyachi et al., Bioorganic & Medicinal Chemistry Letters, vol. 12, No. 1, Jan. 2002, pp. 77-80.
Kurtz, Hcaplus 2006:551484, “New treatment strategies for patients with hypertension and insulin resistance”, American Journal of Medicine, 2006.
Li et al., Hcaplus 2006:256663, “Peroxisome proliferators-activated receptors: how their effects on macrophages can lead to the development of a new drug therapy against atherosclerosis”, Annual Review of Pharmacology and Toxicology, 2006.
Demers et al., Journal of the American Pharmaceutical Association, Scientific Edition, vol. 41, No. 2, 1952, pp. 61-65.
Vasil'eva et al., Database Calpus, “Synthesis and Biological activity of acyl derivatives of 4-aminoantipyrine”, 1984, XP002450796.
Aboul-Enein et al., Database Calpus, “Synthesis and biological activity of dibenz[c,e]azepines”, 1990, XP002450797.
Richter et al., Tetrahedron Letters, vol. 39, 1998, pp. 8747-8750.
Clark Richard
Emori Eita
Harada Hitoshi
Hihara Taro
Inoue Takashi
Birch & Stewart Kolasch & Birch, LLP
Eisai R&D Management Co., Ltd.
Oh Taylor Victor
LandOfFree
Carboxylic acid derivative and salt thereof does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Carboxylic acid derivative and salt thereof, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Carboxylic acid derivative and salt thereof will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-4119813