Carbamoyl substituted heterocycles

Details Carbamoyl substituted heterocycles Carbamoyl substituted heterocycles

1997-05-23

1998-12-15

Fan, Jane

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

5142368, 514318, 544131, 5462714, 546194, C07D41310, A61K 3144

Patent

active

058497668

ABSTRACT:
This invention relates to carbamoyl substituted heterocycles which are .omega.-phenyl-.omega.-(3-pyridyl)-.omega.-alkenoic acid derivatives bearing a carbamoyl substituted oxazolyl or oxazolinyl group on the phenyl ring and which demonstrate utility for thromboxane receptor antagonism and/or thromboxane synthase inhibition, as well as pharmaceutical formulations containing them, methods for their use, and processes and intermediates for their preparation.

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