Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2006-01-31
2006-01-31
Owens, Amelia A. (Department: 1625)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C514S337000, C514S449000, C514S471000, C514S473000, C546S281700, C549S060000, C549S471000, C549S510000, C549S511000
Reexamination Certificate
active
06992104
ABSTRACT:
Taxanes having a carbonate substituent at C(7), a hydroxy substituent at C(10), and a range of C(2), C(9), C(14), and side chain substituents.
REFERENCES:
patent: 5175315 (1992-12-01), Holton
patent: 5227400 (1993-07-01), Holton et al.
patent: 5243045 (1993-09-01), Holton et al.
patent: 5283253 (1994-02-01), Holton et al.
patent: 5319112 (1994-06-01), Kingston et al.
patent: 5350866 (1994-09-01), Holton et al.
patent: 5430160 (1995-07-01), Holton
patent: 5470866 (1995-11-01), Kingston et al.
patent: 5475011 (1995-12-01), Ojima et al.
patent: 5476954 (1995-12-01), Bourzat et al.
patent: 5614645 (1997-03-01), Kingston et al.
patent: 5622986 (1997-04-01), Greenwald et al.
patent: 5698712 (1997-12-01), Bombardelli et al.
patent: 5721268 (1998-02-01), Holton et al.
patent: 5780653 (1998-07-01), Tao et al.
patent: 5811452 (1998-09-01), Ojima et al.
patent: 5824701 (1998-10-01), Greenwald et al.
patent: 5879929 (1999-03-01), Patel
patent: 5912264 (1999-06-01), Wittman et al.
patent: 5939561 (1999-08-01), Bourzat et al.
patent: 5939566 (1999-08-01), Swindell et al.
patent: 5965739 (1999-10-01), Kelly et al.
patent: 0 558 959 (1993-09-01), None
patent: 0 604 910 (1994-07-01), None
patent: 0 629 701 (1994-12-01), None
patent: 0 639 577 (1995-02-01), None
patent: 0 747 385 (2002-08-01), None
patent: WO 93/16059 (1993-08-01), None
patent: WO 94/13655 (1994-06-01), None
patent: WO 95/11241 (1995-04-01), None
patent: WO 96/13495 (1996-05-01), None
patent: WO 96/38138 (1996-12-01), None
patent: WO 97/09979 (1997-03-01), None
patent: WO 97/42181 (1997-11-01), None
patent: WO 99/09021 (1999-02-01), None
patent: WO 01/57013 (2001-08-01), None
Deutsch et al. “Synthesis of Congeners and Prodrugs. 3. Water-Soluble Prodrugs of Taxol with Potent Antitumor Activity” J. Med. Chem., vol. 32, No. 4 (1989) pp. 788-792.
Gueritte-Voegelein et al. “Chemical Studies of 10-Deacetyl Baccatin III. Hemisynthesis of Taxol Derivatives” Tetrahedron Letters, vol. 42, No. 16 (1986) pp. 4451-4460.
Gueritte-Voegelein et al. “Relationships between the Structure of Taxol Analogues and Their Antimitotic Activity” Journal of Medicinal Chemistry, vol. 34, No. 3 (1991) pp. 992-998.
Kant et al. “A Chemoselective Approach to Functionalize the C-10 Position of 10-Deacetylbaccatin III. Synthesis and Biological Properties of Novel C-10 Taxol Analogues” Tetrahedron Letters, vol. 35, No. 30 (1994) pp. 5543-5546.
Ojima et al. “Syntheses and Structure-Activity Relationships of the Second-Generation Antitumor Taxoids: Exceptional Activity Against Drug-Resistant Cancer Cells” Journal of Medicinal Chemistry, vol. 39, No. 20 (1996) pp. 3889-3896.
Ojima et al. “Synthesis of Novel 3′-Trifluoromethyl Taxoids Through Effective Kinetic Resolution of Racemic4-CF3-β-Lactams With Baccatins” CHIRALITY, vol. 9 (1997) pp. 487-494.
Straubinger et al. “Pharmacology and Antitumor Effect of Novel Placlitaxel Formulations” Chapter 8, Edited by G. Georg et al., Taxane Anticancer Agents, Basic Science and Current Status, ACS Symposium Series 583, 207th National Meeting of the American Chemical Society, San Diego, CA (1994) pp. 111-123.
Suffness “Chapter 32. Taxol: From Discovery to Therapeutic Use” Annual Reports in Medicinal Chemistry, vol. 28 (1993) pp. 305-314.
Georgian Search Report from AP 2001 004499 dtd Dec. 25, 2002.
International Search Report for analogous PCT Application No. PCT/US01/03554 dated Jun. 11, 2001.
FSU Research Foundation, Inc.
Owens Amelia A.
Senniger Powers
LandOfFree
C7 carbonate taxane compositions does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with C7 carbonate taxane compositions, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and C7 carbonate taxane compositions will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-3592684