Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2011-08-09
2011-08-09
Fetterolf, Brandon J (Department: 1628)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
active
07994159
ABSTRACT:
It was discovered that a compound represented by the general formula (I) shows strong c-Kit kinase inhibitory activity, and it inhibits proliferation of c-Kit kinase activated-cancer cells in vitro and in vivo. A novel anticancer agent showing c-Kit kinase inhibitory activity was discovered.The general formula (I):(wherein R1represents methyl etc., R2represents cyano etc., R3represents hydrogen etc., R4represents hydrogen etc.).
REFERENCES:
patent: 4526988 (1985-07-01), Hertel et al.
patent: 4742003 (1988-05-01), Derynck et al.
patent: 5180818 (1993-01-01), Cech et al.
patent: 5464826 (1995-11-01), Grindey et al.
patent: 5487889 (1996-01-01), Eckert et al.
patent: 5624937 (1997-04-01), Reel et al.
patent: 5656454 (1997-08-01), Lee et al.
patent: 5658374 (1997-08-01), Glover
patent: 5733913 (1998-03-01), Blankley et al.
patent: 5747651 (1998-05-01), Lemischka
patent: 5750376 (1998-05-01), Weiss et al.
patent: 5770599 (1998-06-01), Gibson
patent: 5792783 (1998-08-01), Tang et al.
patent: 5891996 (1999-04-01), Mateo de Acosta del Rio et al.
patent: 6143764 (2000-11-01), Kubo et al.
patent: 6156522 (2000-12-01), Keay et al.
patent: 6217866 (2001-04-01), Schlessinger et al.
patent: 6346398 (2002-02-01), Pavco et al.
patent: 6476040 (2002-11-01), Norris et al.
patent: 6524583 (2003-02-01), Thorpe et al.
patent: 6534535 (2003-03-01), Zhu et al.
patent: 6676941 (2004-01-01), Thorpe et al.
patent: 6797823 (2004-09-01), Kubo et al.
patent: 6811779 (2004-11-01), Rockwell et al.
patent: 6821987 (2004-11-01), Kubo et al.
patent: 7005430 (2006-02-01), Ueno et al.
patent: 7135466 (2006-11-01), Sakai et al.
patent: 7169789 (2007-01-01), Kubo et al.
patent: 7253286 (2007-08-01), Funahashi et al.
patent: 7435590 (2008-10-01), Komurasaki
patent: 7612092 (2009-11-01), Funahashi et al.
patent: 7612208 (2009-11-01), Matsushima et al.
patent: 2002/0010203 (2002-01-01), Lipson et al.
patent: 2002/0040127 (2002-04-01), Jiang et al.
patent: 2003/0087907 (2003-05-01), Kubo et al.
patent: 2003/0113713 (2003-06-01), Glezer et al.
patent: 2003/0215523 (2003-11-01), Ozawa et al.
patent: 2004/0009965 (2004-01-01), Collins et al.
patent: 2004/0034026 (2004-02-01), Wood et al.
patent: 2004/0053908 (2004-03-01), Funahashi et al.
patent: 2004/0132727 (2004-07-01), Sakai et al.
patent: 2004/0152759 (2004-08-01), Abrams et al.
patent: 2004/0191254 (2004-09-01), Fagin
patent: 2004/0242506 (2004-12-01), Barges Causeret et al.
patent: 2004/0253205 (2004-12-01), Yamamoto et al.
patent: 2005/0014727 (2005-01-01), Muller et al.
patent: 2005/0049264 (2005-03-01), Miwa et al.
patent: 2005/0119303 (2005-06-01), Wakabayashi et al.
patent: 2005/0176802 (2005-08-01), Tang et al.
patent: 2005/0187236 (2005-08-01), Tsuruoka et al.
patent: 2005/0272688 (2005-12-01), Higgins et al.
patent: 2005/0277652 (2005-12-01), Matsushima et al.
patent: 2006/0004017 (2006-01-01), Stokes et al.
patent: 2006/0004029 (2006-01-01), Tsuruoka et al.
patent: 2006/0057195 (2006-03-01), Nonomura et al.
patent: 2006/0079494 (2006-04-01), Santi et al.
patent: 2006/0135486 (2006-06-01), Owa et al.
patent: 2007/0004773 (2007-01-01), Sakaguchi et al.
patent: 2007/0027318 (2007-02-01), Kubo et al.
patent: 2007/0032521 (2007-02-01), Moussy et al.
patent: 2007/0037849 (2007-02-01), Naito et al.
patent: 2007/0078159 (2007-04-01), Matsushima
patent: 2007/0117842 (2007-05-01), Arimoto et al.
patent: 2008/0214604 (2008-09-01), Furitsu et al.
patent: 2009/0047278 (2009-02-01), Owa et al.
patent: 2009/0047365 (2009-02-01), Owa et al.
patent: 203126 (1986-06-01), None
patent: 0 602 851 (1996-10-01), None
patent: 0 795 556 (1997-09-01), None
patent: 0 837 063 (1998-04-01), None
patent: 0 405 425 (1998-08-01), None
patent: 0 870 842 (1998-10-01), None
patent: 0 684 820 (2001-08-01), None
patent: 1 153 920 (2001-11-01), None
patent: 0712863 (2002-02-01), None
patent: 1 029 853 (2004-02-01), None
patent: 1415987 (2004-05-01), None
patent: 1522540 (2005-04-01), None
patent: 1535910 (2005-06-01), None
patent: 1566379 (2005-08-01), None
patent: 1604665 (2005-12-01), None
patent: 1 683 785 (2006-07-01), None
patent: 1 698 623 (2006-09-01), None
patent: 1698623 (2006-09-01), None
patent: 1859797 (2007-11-01), None
patent: 1925676 (2008-05-01), None
patent: 1925941 (2008-05-01), None
patent: 1949902 (2008-07-01), None
patent: 1964837 (2008-09-01), None
patent: 1 797 881 (2009-04-01), None
patent: 2 253 848 (1992-09-01), None
patent: 63-028427 (1988-02-01), None
patent: 1022874 (1989-01-01), None
patent: 02-291295 (1990-12-01), None
patent: 4341454 (1992-11-01), None
patent: 06-153952 (1994-06-01), None
patent: 7-176103 (1995-07-01), None
patent: 8-045927 (1996-02-01), None
patent: H8-048078 (1996-02-01), None
patent: 09-023885 (1997-01-01), None
patent: 09-234074 (1997-09-01), None
patent: 11-501343 (1999-02-01), None
patent: 11-143429 (1999-05-01), None
patent: 11-158149 (1999-06-01), None
patent: 11-322596 (1999-11-01), None
patent: 3040486 (2000-03-01), None
patent: 3088018 (2000-07-01), None
patent: 2000-328080 (2000-11-01), None
patent: 2001-131071 (2001-05-01), None
patent: 2002-003365 (2002-01-01), None
patent: 2002-114710 (2002-04-01), None
patent: 2002-536414 (2002-10-01), None
patent: 2003-012668 (2003-01-01), None
patent: 2003-026576 (2003-01-01), None
patent: 3420549 (2003-04-01), None
patent: 2003-525595 (2003-09-01), None
patent: 2004-513964 (2004-05-01), None
patent: 2004-155773 (2004-06-01), None
patent: 2004-531549 (2004-10-01), None
patent: 2005-501074 (2005-01-01), None
patent: 2005-504111 (2005-02-01), None
patent: 2005-520834 (2005-07-01), None
patent: 3712393 (2005-08-01), None
patent: 2006-508981 (2006-03-01), None
patent: 2006-515884 (2006-06-01), None
patent: 86/03222 (1986-06-01), None
patent: WO 92/20642 (1992-11-01), None
patent: WO 95/15758 (1995-06-01), None
patent: WO 95/19774 (1995-07-01), None
patent: WO 96/09294 (1996-03-01), None
patent: WO 96/26997 (1996-09-01), None
patent: 96/30347 (1996-10-01), None
patent: 96/33980 (1996-10-01), None
patent: WO 96/39145 (1996-12-01), None
patent: WO 96/40142 (1996-12-01), None
patent: WO 97/03069 (1997-01-01), None
patent: WO 97/13760 (1997-04-01), None
patent: WO 97/13771 (1997-04-01), None
patent: 97/17329 (1997-05-01), None
patent: WO 97/21437 (1997-06-01), None
patent: WO 97/38984 (1997-10-01), None
patent: 97/48693 (1997-12-01), None
patent: WO 98/00134 (1998-01-01), None
patent: WO 98/02434 (1998-01-01), None
patent: WO 98/02437 (1998-01-01), None
patent: WO 98/02438 (1998-01-01), None
patent: 98/14437 (1998-04-01), None
patent: WO 98/13350 (1998-04-01), None
patent: WO 98/23613 (1998-06-01), None
patent: WO 98/32436 (1998-07-01), None
patent: 98/35958 (1998-08-01), None
patent: WO 98/37079 (1998-08-01), None
patent: WO 98/50346 (1998-11-01), None
patent: WO 98/52558 (1998-11-01), None
patent: WO 99/00357 (1999-01-01), None
patent: 99/35146 (1999-07-01), None
patent: WO 99/32106 (1999-07-01), None
patent: WO 99/32110 (1999-07-01), None
patent: WO 99/32111 (1999-07-01), None
patent: WO 99/32436 (1999-07-01), None
patent: WO 99/35132 (1999-07-01), None
patent: WO 99/43654 (1999-09-01), None
patent: 99/62890 (1999-12-01), None
patent: 00/31048 (2000-06-01), None
patent: 00/42012 (2000-07-01), None
patent: 00/43366 (2000-07-01), None
patent: WO 00/42012 (2000-07-01), None
patent: WO 00/43384 (2000-07-01), None
patent: 00/47212 (2000-08-01), None
patent: WO 00/44728 (2000-08-01), None
patent: WO 00/47212 (2000-08-01), None
patent: WO 00/50405 (2000-08-01), None
patent: WO 00/71097 (2000-11-01), None
patent: 01/02369 (2001-01-01), None
patent: 01/23375 (2001-04-01), None
patent: 01/27081 (2001-04-01), None
patent: 01/32926 (2001-05-01), None
patent: WO-01/36403 (2001-05-01), None
patent: 01/40217 (2001-06-01), None
patent: WO 01/45689 (2001-06-01), None
patent: 01/47890 (2001-07-01), None
patent: 01/47931 (2001-07-01), None
patent: 01/60814 (2001-08-01), None
patent: WO 02/16348 (2002-02-01), None
patent: 02/32872 (2002-04-01), None
patent: 02/36117 (2002-05-01), None
patent: 02/41882 (2002-05-01), None
patent: 02/072578 (2002-09-01), None
patent: WO 02/72578 (2002-09-01), None
patent: 02/080975 (2002
Okada Masayuki
Tsuruoka Akihiko
Watanabe Tatsuo
Yamamoto Yuji
EISAI R&D Management Co., Ltd.
Fetterolf Brandon J
Fish & Richardson P.C.
Pagonakis Anna
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