Boronated phosphoramidate compounds

Chemistry: natural resins or derivatives; peptides or proteins; – Peptides of 3 to 100 amino acid residues

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530324, 530325, 530326, 530327, 530328, 530329, 530330, 530331, 530350, 536 221, 536 255, 536 264, 536 245, 536 2644, 536 267, 536 268, 558 72, C07K 504, C07K 704, C07F 902, A61K 3702

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active

052722503

ABSTRACT:
A class of pharmaceutically active boronated compounds are provided. The boronated compounds include boronated phosphoramidates, and boronated nucleosides, and oligomers thereof. The compounds are boronated by an aminoalkyl substituted polyborane, carborane, metallopolyborane or metallocarborane.

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