Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1988-04-08
1990-12-11
Springer, David B.
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
556 7, C07C10352, C07C 502
Patent
active
049772686
ABSTRACT:
Novel boron dipeptide analogs and their corresponding amide derivatives which exhibit significant antihyperlipidemic and antineoplastic activities. Methods for preparing the boron containing compounds are disclosed as well as methods for utilizing the compounds to induce antihyperlipidemic and antineoplastic activity.
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Spielvogel, Das, McPhail, Onan and Hall, "Boron Analogues of the a-Amino Acids, Synthesis, X-ray Crystal Structure, and Biological Activity of Ammonia-Carboxyborane, the Boron Analogue of Glycine", Journal of the American Chemical Society, 1980, pp. 6343-6343.
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Hall Iris H.
McPhail Andrew T.
Spielvogel Bernard F.
Duke University
Jenkins Richard E.
Springer David B.
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