Bis-sulfonamide hydroxyethylamino retroviral protease...

Details Bis-sulfonamide hydroxyethylamino retroviral protease... Bis-sulfonamide hydroxyethylamino retroviral protease...

2007-11-20

2007-11-20

Stockton, Laura L. (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Four or more ring nitrogens in the bicyclo ring system

C544S360000, C544S383000, C546S247000

Reexamination Certificate

active

11349352

ABSTRACT:
Bis-sulfonamido hydroxyethylamino compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to retroviral protease inhibiting compounds of the formula:or a pharmaceutically acceptable salt, prodrug or ester thereof, wherein the variables are as defined herein.

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