Bis-piperidinyl non-peptidyl neurokinin receptor antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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Details

546187, A61K 31445, C07D40114

Patent

active

055300090

ABSTRACT:
This invention provides novel compound of the formula ##STR1## which is neurokinin receptor antagonist.

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Hispskind et al. "Pharmacological characterization of LY 303870: a novel potent and selective nonpeptide substance P receptor antagonist" Pharmcol. Exp. Ther. v. 275, pp. 737-744 (1995).

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