Bis-amino acid hydroxyethylamino sulfonamide retroviral...

Details Bis-amino acid hydroxyethylamino sulfonamide retroviral... Bis-amino acid hydroxyethylamino sulfonamide retroviral...

2006-08-10

2008-03-04

Kumar, Shailendra (Department: 1621)

Organic compounds -- part of the class 532-570 series

Organic compounds

Amino nitrogen containing

C514S311000, C514S367000, C514S394000, C514S456000, C514S464000, C514S467000, C514S487000, C514S602000, C514S604000, C549S366000, C549S434000, C549S437000, C549S438000, C549S443000, C549S467000

Reexamination Certificate

active

07339078

ABSTRACT:
Selected bis-amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to such retroviral protease inhibitors and, more particularly, relates to selected novel compounds, compositions, and methods for inhibiting retroviral proteases, such as human immunodeficiency virus (HIV) protease, prophylactically preventing retroviral infection or the spread of a retrovirus, and treatment of a retroviral infection.

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