Biotinylated small molecules

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

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435 5, 435 6, 435 9, 436804, 436808, 436544, 436545, 534 14, 534 15, A61K 4300, A61K 4902, C07D23500, C07D49504

Patent

active

052833429

ABSTRACT:
Methods, compounds, compositions and kits that relate to pretargeted delivery of diagnostic and therapeutic agents are disclosed. In particular, methods for radiometal labeling of biotin and for improved radiohalogenation of biotin, as well as related compounds, are described.

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