Biologically active 1-thio derivatives of vitamin D

Details Biologically active 1-thio derivatives of vitamin D Biologically active 1-thio derivatives of vitamin D

1985-03-18

1987-04-28

Schenkman, Leonard

Chemistry of carbon compounds

Miscellaneous organic carbon compounds

C-metal

C07J 900, A61K 3159

Patent

active

046612947

ABSTRACT:
Novel synthetic derivatives of vitamin D compounds are disclosed as well as processes for their synthesis. The novel compounds are 1-alpha-thio and acylated, 1-beta-thio derivatives of vitamin D compounds and the glycosylated, hydroxylated, fluorinated, and glycosylated orthoester analogues thereof.

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