Bicyclic heterocycles, drugs containing said compounds, use...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S212010, C514S266400, C540S484000, C544S293000, C544S358000

Reexamination Certificate

active

07998949

ABSTRACT:
The present invention relates to bicyclic heterocycles of general formulawhereinRa, Rband Rcare defined as in claim1, their tautomers, their stereoisomers, their mixtures and their salts, in particular their physiologically acceptable salts with inorganic or organic acids and bases, which have valuable pharmacological properties, in particular an inhibitory action on the signal transduction mediated by tyrosine kinases, their use for the treatment of illnesses, in particular of tumoral diseases and of benign prostatic hyperplasia (BPH), of diseases of the lung and of the airways, and the preparation thereof.

REFERENCES:
patent: 3985749 (1976-10-01), Foster
patent: 4322420 (1982-03-01), Kobayashi et al.
patent: 4335127 (1982-06-01), Vandenberk et al.
patent: 4640920 (1987-02-01), Boyle et al.
patent: 4845629 (1989-07-01), Murga
patent: 4921863 (1990-05-01), Sugimoto et al.
patent: 5064833 (1991-11-01), Ife et al.
patent: 5252586 (1993-10-01), Cain et al.
patent: 5457105 (1995-10-01), Barker
patent: 5616582 (1997-04-01), Barker
patent: 5642285 (1997-06-01), Woo et al.
patent: 5721237 (1998-02-01), Myers et al.
patent: 5747498 (1998-05-01), Schnur et al.
patent: 5760041 (1998-06-01), Wissner et al.
patent: 5770599 (1998-06-01), Gibson
patent: 5770603 (1998-06-01), Gibson
patent: 5821246 (1998-10-01), Brown et al.
patent: 5866572 (1999-02-01), Barker et al.
patent: 5929080 (1999-07-01), Frost
patent: 5938706 (1999-08-01), Feldman
patent: 5962458 (1999-10-01), Lohmann et al.
patent: 6004967 (1999-12-01), McMahon et al.
patent: 6046206 (2000-04-01), Pamukcu et al.
patent: 6117433 (2000-09-01), Edens et al.
patent: 6126917 (2000-10-01), Mishani et al.
patent: 6177433 (2001-01-01), Uckun et al.
patent: 6225318 (2001-05-01), Sobolov-Jaynes et al.
patent: 6270747 (2001-08-01), Nadel et al.
patent: 6297258 (2001-10-01), Wissner et al.
patent: 6313130 (2001-11-01), Uckun et al.
patent: 6326373 (2001-12-01), Uckun et al.
patent: 6362336 (2002-03-01), Lohmann et al.
patent: 6384223 (2002-05-01), Gletsos
patent: 6399602 (2002-06-01), Barker et al.
patent: 6403580 (2002-06-01), Himmelsbach et al.
patent: 6414148 (2002-07-01), Thomas et al.
patent: 6551989 (2003-04-01), Nadel et al.
patent: 6562319 (2003-05-01), Mishani et al.
patent: 6566324 (2003-05-01), Nadel et al.
patent: 6617329 (2003-09-01), Himmelsbach et al.
patent: 6627634 (2003-09-01), Himmelsbach et al.
patent: 6645969 (2003-11-01), Myers et al.
patent: 6653305 (2003-11-01), Himmelsbach et al.
patent: 6656946 (2003-12-01), Himmelsbach et al.
patent: 6740561 (2004-05-01), Himmelsbach et al.
patent: 6846799 (2005-01-01), Nadel et al.
patent: 6924285 (2005-08-01), Himmelsbach et al.
patent: 6972288 (2005-12-01), Himmelsbach et al.
patent: 7081461 (2006-07-01), Mortlock et al.
patent: 7119084 (2006-10-01), Himmelsbach et al.
patent: 7196091 (2007-03-01), Himmelsbach et al.
patent: 7354894 (2008-04-01), Nadel et al.
patent: 7358222 (2008-04-01), Nadel et al.
patent: 7456189 (2008-11-01), Himmelsbach et al.
patent: 7531500 (2009-05-01), Nadel et al.
patent: 7700547 (2010-04-01), Nadel et al.
patent: 2001/0036919 (2001-11-01), Nadel et al.
patent: 2001/0041178 (2001-11-01), Nadel et al.
patent: 2001/0044435 (2001-11-01), Himmelsbach et al.
patent: 2002/0049197 (2002-04-01), Himmelsbach et al.
patent: 2002/0082270 (2002-06-01), Himmelsbach et al.
patent: 2002/0082271 (2002-06-01), Himmelsbach et al.
patent: 2002/0115675 (2002-08-01), Himmelsbach et al.
patent: 2002/0128553 (2002-09-01), Mishani et al.
patent: 2002/0169180 (2002-11-01), Himmelsbach et al.
patent: 2002/0173509 (2002-11-01), Himmelsbach et al.
patent: 2002/0173646 (2002-11-01), Thomas et al.
patent: 2002/0177601 (2002-11-01), Himmelsbach et al.
patent: 2003/0148990 (2003-08-01), Nadel et al.
patent: 2003/0149062 (2003-08-01), Jung et al.
patent: 2003/0158196 (2003-08-01), Jung et al.
patent: 2004/0044014 (2004-03-01), Himmelsbach et al.
patent: 2004/0048880 (2004-03-01), Himmelsbach et al.
patent: 2004/0176361 (2004-09-01), Fujio et al.
patent: 2004/0265302 (2004-12-01), Nadel et al.
patent: 2005/0014772 (2005-01-01), Himmelsbach et al.
patent: 2005/0059661 (2005-03-01), Jung et al.
patent: 2005/0070560 (2005-03-01), Himmelsbach et al.
patent: 2005/0159436 (2005-07-01), Himmelsbach et al.
patent: 2005/0165035 (2005-07-01), Bradbury et al.
patent: 2005/0182043 (2005-08-01), Himmelsbach et al.
patent: 2005/0215574 (2005-09-01), Bradbury et al.
patent: 2006/0063752 (2006-03-01), Himmelsbach et al.
patent: 2006/0264450 (2006-11-01), Himmelsbach et al.
patent: 2006/0270672 (2006-11-01), Himmelsbach et al.
patent: 2007/0135463 (2007-06-01), Himmelsbach et al.
patent: 2007/0270330 (2007-11-01), Nadel et al.
patent: 2008/0103161 (2008-05-01), Himmelsbach et al.
patent: 2008/0175797 (2008-07-01), Nadel et al.
patent: 2008/0199462 (2008-08-01), Nadel et al.
patent: 2009/0036676 (2009-02-01), Himmelsbach et al.
patent: 2009/0203683 (2009-08-01), Himmelsbach et al.
patent: 2009/0306072 (2009-12-01), Jung et al.
patent: 2417897 (2003-01-01), None
patent: 2 476 008 (2003-10-01), None
patent: 2 631 813 (2007-06-01), None
patent: 2669187 (2008-05-01), None
patent: 10042058 (2002-03-01), None
patent: 288563 (1988-11-01), None
patent: 326330 (1989-08-01), None
patent: 520722 (1992-12-01), None
patent: 0566226 (1993-10-01), None
patent: 607439 (1994-07-01), None
patent: 635507 (1995-01-01), None
patent: 0787722 (1997-08-01), None
patent: 837063 (1998-04-01), None
patent: 1230919 (2002-08-01), None
patent: 1283039 (2003-02-01), None
patent: 1369418 (2003-12-01), None
patent: 2033894 (1980-05-01), None
patent: 2160201 (1985-12-01), None
patent: 2295387 (1996-05-01), None
patent: 11-189586 (1999-07-01), None
patent: 88/02365 (1988-04-01), None
patent: 92/14746 (1992-09-01), None
patent: 92/20642 (1992-11-01), None
patent: 93/08170 (1993-04-01), None
patent: 93/17682 (1993-09-01), None
patent: 602851 (1994-06-01), None
patent: 94/27965 (1994-12-01), None
patent: 95/00146 (1995-01-01), None
patent: 95/03283 (1995-02-01), None
patent: 95/15758 (1995-06-01), None
patent: 95/19169 (1995-07-01), None
patent: 95/24190 (1995-09-01), None
patent: 96/09294 (1996-03-01), None
patent: 96/15118 (1996-05-01), None
patent: 96/16960 (1996-06-01), None
patent: 96/30347 (1996-10-01), None
patent: 96/33977 (1996-10-01), None
patent: 96/33978 (1996-10-01), None
patent: 96/33979 (1996-10-01), None
patent: 96/33980 (1996-10-01), None
patent: 96/33981 (1996-10-01), None
patent: 96/39145 (1996-12-01), None
patent: 97/03069 (1997-01-01), None
patent: 97/11692 (1997-04-01), None
patent: 97/18813 (1997-05-01), None
patent: 97/22596 (1997-06-01), None
patent: 97/30034 (1997-08-01), None
patent: 97/30035 (1997-08-01), None
patent: 97/30044 (1997-08-01), None
patent: 97/32856 (1997-09-01), None
patent: 97/38983 (1997-10-01), None
patent: 97/38994 (1997-10-01), None
patent: 97/42187 (1997-11-01), None
patent: 98/02434 (1998-01-01), None
patent: 98/13354 (1998-04-01), None
patent: 98/19649 (1998-05-01), None
patent: 98/38984 (1998-09-01), None
patent: 98/43960 (1998-10-01), None
patent: 98/50038 (1998-11-01), None
patent: 98/50370 (1998-11-01), None
patent: 99/01467 (1999-01-01), None
patent: 99/06378 (1999-02-01), None
patent: 99/06396 (1999-02-01), None
patent: 99/09016 (1999-02-01), None
patent: 99/10349 (1999-03-01), None
patent: 99/24037 (1999-05-01), None
patent: 99/35132 (1999-07-01), None
patent: 99/61428 (1999-12-01), None
patent: 00/00202 (2000-01-01), None
patent: 00/06555 (2000-02-01), None
patent: 00/09481 (2000-02-01), None
patent: 00/10981 (2000-03-01), None
patent: 00/12497 (2000-03-01), None
patent: 00/18740 (2000-04-01), None
patent: 00/20402 (2000-04-01), None
patent: 00/24718 (2000-05-01), None
patent: 00/44728 (2000-08-01), None
patent: 00/47212 (2000-08-01), None
patent: 00/51587 (2000-09-01), None
patent: 00/51991 (2000-09-01), None
patent: 00/55141 (2000-09-01), None
patent: 00/55162 (2000-09-01), None
patent: 00/56338 (2000-09-01), None
patent: 00/56720 (2000-09-01), None
patent: 00/68201 (2000-11-01), None
patent: 00/68203 (2000-11-01), None
patent: 00/73260 (2000-12-01), None
patent: 00/78735 (2000-12

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