Bicyclic derivatives for use in the treatment of androgen...

Details Bicyclic derivatives for use in the treatment of androgen... Bicyclic derivatives for use in the treatment of androgen...

2011-08-23

2011-08-23

Hui, San-Ming (Department: 1628)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C514S360000, C514S383000, C544S236000, C548S262400

Reexamination Certificate

active

08003649

ABSTRACT:
The invention concerns bicyclic compounds of Formula Iwherein the integers X1, X2, X3, Ring A, R4, R5and m are as defined in the description. The present invention also relates to processes for the preparation of such compounds, pharmaceutical compositions containing them and their use in the manufacture of a medicament for use in the prevention or treatment of androgen-receptor associated conditions.

REFERENCES:
patent: 2006039325 (2006-04-01), None
patent: 2008109104 (2008-09-01), None
RN 334500-45-7 Registry file of chemical abstract services entered STN on May 3, 2001.
RN 927049-23-8 Registry file of chemical abstract services entered STN on Mar. 18, 2007.
RN 930466-59-4 Registry file of chemical abstract services entered STN on Apr. 17, 2007.
RN 930503-83-6 Registry file of chemical abstract services entered STN on Apr. 17, 2007.
RN 931060-90-1 Registry file of chemical abstract services entered STN on Apr. 19, 2007.
Bioorg. Med. Chem. Lett. 2007; vol. 17; Issue 16, pp. 4579-4583.
Sep. 23, 2008 Novelty Search Results.
Vasaitis et. al. Androgen receptor inactivation contributes to antitumor efficacy of 17 -hydroxylase/17,20-lyase inhibitor 3 -hydroxy-17-(1H-benzimidazole-1-yl)androsta-5, 16-diene in prostate cancer; Molecular Cancer Therapeutics 2008;7(8). Aug. 2008; pp. 2348-2357.

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