Bicyclic .beta.-lactam antibiotics

Details Bicyclic .beta.-lactam antibiotics Bicyclic .beta.-lactam antibiotics

1993-02-24

1995-02-28

Rizzo, Nicholas

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D48704

Patent

active

053938828

ABSTRACT:
A method for preparing 2-amino-.beta.-lactams which are substituted by readily-removed protecting groups is provided. According to this invention, an acyl-2-amino-.beta.-lactam is further acylated with a different acyl group and is subsequently treated with base to provide a protected 2-amino .beta.-lactam with a more desirable protecting group.

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Spry, Heterocycles, 26, 2911 (1987).

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