Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2005-11-15
2005-11-15
Dentz, Bernard (Department: 1625)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C514S311000, C514S313000, C546S155000, C546S157000, C546S159000, C546S160000, C546S171000, C546S172000, C546S173000
Reexamination Certificate
active
06964973
ABSTRACT:
The present invention is directed to compounds, pharmaceutical compositions, and methods for modulating processes mediated by AR and PR. More particularly, the invention relates to nonsteroidal compounds and compositions that are high affinity, high specificity agonists, partial agonists (i.e., partial activators and/or tissue-specific activators) and antagonists for AR and PR. Also provided are methods of making such compounds and pharmaceutical compositions, as well as critical intermediates used in their synthesis.
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Farmer Luc
Pio Barbara
Zhi Lin
Dentz Bernard
Fish & Richardson P.C.
Ligand Pharmaceuticals Incorporated
Miskiel Frank J.
Seidman Stephanie L.
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