Organic compounds -- part of the class 532-570 series – Organic compounds – Four or more ring nitrogens in the bicyclo ring system
Reexamination Certificate
2003-05-30
2010-02-16
Wilson, James O (Department: 1624)
Organic compounds -- part of the class 532-570 series
Organic compounds
Four or more ring nitrogens in the bicyclo ring system
Reexamination Certificate
active
07662960
ABSTRACT:
Conformationally constrained compounds of structure:which mimic the secondary structure of β-strand regions of biologically active peptides and proteins are disclosed. Such β-strand mimetic structures have utility over a wide range of fields, including use as diagnostic and therapeutic agents that inhibit protease, kinase and the like. Libraries containing the β-strand mimetic structures of this invention are also disclosed as well as methods for screening the same to identify biologically active members.
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Chung Jae Uk
Eguchi Masakatsu
Kahn Michael
Moon Sung Hwan
Choongwae Pharma Corporation
Murray Jeffrey H
SEED Intellectual Property Law Group PLLC
Wilson James O
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