Benzoyl- and .alpha.-hydroxybenzyl-phenyl-glycosides and applica

Drug – bio-affecting and body treating compositions – Conjugate or complex of monoclonal or polyclonal antibody,... – Conjugated via claimed linking group – bond – chelating agent,...

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536 41, 536 179, 536 176, 536 178, A61K 3170, C07H 1520

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active

044329733

ABSTRACT:
The present invention relates to the benzoyl- and .alpha.-hydroxybenzyl-phenyl-oside derivatives of general formula: ##STR1## [in which Z is CO or CHOH, X.sub.1, X.sub.2, X.sub.3, X.sub.4 and X.sub.5, which are identical or different, each represent an atom of hydrogen, an atom of halogen, an alkyl group with 1 to 4 carbon atoms, an alkyl group with 1 to 4 carbon atoms substituted by one or more atoms of halogen, an OH group, an alkoxy group with 1 to 4 carbon atoms, an alkoxy group with 1 to 4 carbon atoms, substituted by one or more atoms of halogen, a nitro group, a cyano group, a thiocyano group, an isothiocyano group, a NR'R" group (where R' and R", identical or different, each represent an atom of hydrogen or an alkyl group with 1 to 4 carbon atoms) X.sub.1 being able, in addition, to represent an --NH--CS--O--CH.sub.3 group or an --O--C(CH.sub.3).sub.2 CO.sub.2 --R'" group (where R'" is an alkyl group with 1 to 4 carbon atoms and, preferably, an isopropyl group); and R represents a radical ose (the hydroxyl and amine functions of the radical ose being able to be substituted by acyl, alkyl or sulfate groups)], and to their diastereoisomers. It also relates to the method for preparing these derivatives and to their application in therapeutics.

REFERENCES:
patent: 2218569 (1940-10-01), White
patent: 2798079 (1957-07-01), Linn
patent: 3152115 (1964-10-01), Morel et al.
patent: 3356674 (1967-12-01), Ikeda et al.
patent: 3496196 (1970-02-01), Suami et al.
patent: 3960835 (1976-06-01), Robertson

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