Benzoxepins as intermediates to 5HT.sub.3 antagonists

Details Benzoxepins as intermediates to 5HT.sub.3 antagonists Benzoxepins as intermediates to 5HT.sub.3 antagonists

1989-07-31

1990-05-08

Schwartz, Richard A.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D31308

Patent

active

049240102

ABSTRACT:
Certain specific substituted 9-N-(1-azabicycolo-[2.2.2.]octan-3-yl)carboxamido-2,3,4,5-tetrahydro-1-ben zoxepins and their valuable use as 5-HT.sub.3 antagonists having CNS and gastric prokinetic activity and void of any significant D.sub.2 receptor binding properties are disclosed. Methods for their preparation also are described.

REFERENCES:
patent: 4332039 (1980-11-01), Closse et al.
Christensen, H. Synthetic Communications 4(1) 1974, pp. 1-9.

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