Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2006-01-31
2006-01-31
Solola, Taofiq (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S338000, C514S377000, C514S422000, C544S138000, C546S269100, C548S222000, C548S518000, C549S414000
Reexamination Certificate
active
06992083
ABSTRACT:
The invention relates to compounds of formulawhereinR is phenyl, unsubstituted or substituted by halogen or —CH2N(CH3)(CH2)nOCH3, oris benzyl,lower alkyl,lower alkoxy,—(CH2)nOCH3, or ispyridin 3 -or 4-yl, unsubstituted or substituted by lower alkyl, halogen, morpholinyl, —(CH2)n-halogen, —(CH2)nOCH3, —(CH2)n-morpholin-4-yl, or —(CH2)n-pyrrolidin-1-yl;R1is phenyl, unsubstituted or substituted by halogen,tetrahydropyran-4-yl, 3,6-dihydro-2H-pyran-4-yl or morpholin-4-yl;n is independently from each other 1 or 2;and to pharmaceutically acceptable salts thereof for the treatment of diseases related to the adenosine A2A-receptor.
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Hoffman-La Roche Inc.
Johnston George W.
Lee Susannah E.
Prior Kimberly J.
Rocha-Tramaloni Patricia S.
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