Benzoxazepinone derivatives

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C540S490000

Reexamination Certificate

active

07060698

ABSTRACT:
The invention relates to benzoxazepinone derivatives of formulawhereinR1, R2, R3, R4, and n are as defined in the specification and to a pharmaceutically suitable acid addition salt thereof. These compounds are good γ-secretase inhibitors for the treatment of Alzheimer's disease.

REFERENCES:
patent: WO 01/98282 (2001-12-01), None
patent: WO 02/30912 (2002-04-01), None
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Brockhaus, M. et al., Neuroreport vol. 9(7), 1998, pp. 1481-1486.

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