Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1998-09-22
2000-05-09
Chang, Ceila
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
5142335, 514253, 514307, 514422, 514443, 544146, 544376, 546202, 546237, 548525, 548527, 549 51, A61K 31445, C07D40908
Patent
active
060604883
ABSTRACT:
This invention is related to novel benzothiophene compounds of formula I: ##STR1## where R, R.sup.1, R.sup.2, X and m are as defined in the specification, which are useful for the inhibition of the various medical conditions associated with postmenopausal syndrome, as well as estrogen dependent diseases including cancer of the breast, uterus, and cervix. The present invention further relates to pharmaceutical formulations of compounds of formula I.
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Dodge Jeffrey Alan
Stocksdale Mark Gregory
Chang Ceila
Eli Lilly and Company
Voy Gilbert T.
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