Benzothiepines having activity as inhibitors of ileal bile acid

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514336, 514382, 514397, 549 9, 5462797, 548252, 5483151, A61K 3138, A61K 3144, C07D33700, C07D21172

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active

059943912

ABSTRACT:
Provided are novel benzothiepines, derivatives, and analogs thereof; pharmaceutical compositions containing them; and methods of using these compounds and compositions in medicine, particularly in the prophylaxis and treatment of hyperlipidemic conditions such as those associated with atherosclerosis or hypercholesterolemia, in mammals.

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