Benzothiazin and benzoxazin derivatives; their preparation and u

Details Benzothiazin and benzoxazin derivatives; their preparation and u Benzothiazin and benzoxazin derivatives; their preparation and u

1998-10-26

2000-10-10

Raymond, Richard L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

5142305, 544 50, 544 92, A61K 3154, A61K 31535, C07D27916, C07D26512

Patent

active

061302147

ABSTRACT:
The present invention relates to novel antiobesity and hypocholesterolemic compounds, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and pharmaceutically acceptable compositions containing them. More particularly, the present invention relates to novel .beta.-aryl-.alpha.-oxysubstituted alkylcarboxylic acids of the general formula (I), their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and pharmaceutically acceptable compositions containing them. ##STR1##

REFERENCES:
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Buckle, D.R. "Non Thiazolidinedione Antihyperglyceaemic Agents . . . " Bioorganic & Medicinal Chemistry Letters, vol. 6, No. 17, pp. 2121-2126, 1996.
Hulin, B. "Hypoglycemic Activity of A Series of . . . " J. Med. Chem. 36, 1996, pp. 3897-3907.
Patent Abstracts of Japan vol. 97, No. 5, May 30, 1997 & JP 09 012575, Jan. 14, 1997.
Patent Abstracts of Japan vol. 17, No. 627 (C11-31) Nov. 19, 1993 & JP 05 194236A.

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