Benzopyran-containing compounds and method for their use

Details Benzopyran-containing compounds and method for their use Benzopyran-containing compounds and method for their use

1995-02-21

2000-05-09

Criares, Theodore J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514320, 514337, 514345, A61K 3140, A61K 3144

Patent

active

060605030

ABSTRACT:
Certain benzopyran antiestrogens are disclosed for treating estrogen sensitive diseases such as breast cancer. Prodrug forms provide ease of manufacturing, good shelf life, and bioavailability, and preferred stereoisomers are shown to be more effective than racemic mixtures.

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