Benzoindoline compounds

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C544S372000

Reexamination Certificate

active

06998403

ABSTRACT:
A compound of formula (I):wherein:R1and R2together form a benzo ring optionally substituted by halogen or by alkyl, alkoxy, cyano, nitro, hydroxy, amino, alkylamino, dialkylamino or trifluoromethyl, and R3and R4represent hydrogen,orR1and R4represent hydrogen and R2and R3together form a benzo ring optionally substituted by halogen or by alkyl, alkoxy, cyano, nitro, hydroxy, amino, alkylamino, dialkylamino or trifluoromethyl,orR1and R2represent hydrogen and R3and R4together form a benzo ring optionally substituted by halogen or by alkyl, alkoxy, cyano, nitro, hydroxy, amino, alkylamino, dialkylamino or trifluoromethyl,addition salts thereof with a pharmaceutically acceptable acid or base, andmethods of treating conditions susceptible to α2-AR/5-HT2Cantagonists.

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