Benzodiazepine derivatives

Details Benzodiazepine derivatives Benzodiazepine derivatives

1975-06-23

1977-09-06

Jiles, Henry R.

Drug, bio-affecting and body treating compositions

Antigen, epitope, or other immunospecific immunoeffector

Bacterium or component thereof or substance produced by said...

2602393D, 260562N, 260562B, 260570AB, C07D24324

Patent

active

040468909

ABSTRACT:
This invention is directed to pharmacologically active compounds of the formula ##STR1## wherein R.sub.1 represents a hydrogen atom or lower alkyl group and R.sub.2 represents a halogen atom.
The compounds of formula I are optically active and have the absolute configuration S at the carbon atom in the 3-position. They exhibit anthelmintic, sedative, anticonvulsant and muscle relaxant activity.
Also provided are methods for their preparation and formulations which incorporate the active compounds.

REFERENCES:
patent: 3116203 (1963-12-01), Kariss et al.
patent: 3121076 (1964-02-01), Keller et al.
patent: 3123529 (1964-03-01), Kariss et al.
patent: 3248223 (1966-04-01), Bauernfeind
patent: 3998811 (1976-12-01), Kajfez et al.
Sunjic et al., "J. Het. Chem." vol. 10 (1973) pp. 591-599.
Stempel et al., "J. Org. Chem." vol. 27 (1962) pp. 4675-4677.

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