Benzimidazolidinone derivatives as muscarinic agents

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C514S216000, C514S217100, C514S304000, C514S321000, C548S321500, C548S152000, C548S217000, C548S304700, C548S465000

Reexamination Certificate

active

11418340

ABSTRACT:
Benzimidazolidinone derivative compounds, which increase acetylcholine signaling or effect in the brain, and highly selective muscarinic agonists, particularly for the M1and/or M4receptor subtypes, pharmaceutical compositions comprising the same, as well as methods of treating psychosis using these compounds are disclosed.

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