Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2011-03-15
2011-03-15
Stockton, Laura L. (Department: 1626)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C514S394000
Reexamination Certificate
active
07906654
ABSTRACT:
Provided herein are compounds in accord with Formula I:that are useful in the treatment of pain.
REFERENCES:
patent: 3624103 (1971-11-01), De Martiis et al.
patent: 3839347 (1974-10-01), Fisher et al.
patent: 4722929 (1988-02-01), Austel et al.
patent: 4738981 (1988-04-01), Horwell
patent: 6794404 (2004-09-01), Beaulieu et al.
patent: 2003/0149050 (2003-08-01), Jagtap et al.
patent: 2003/0158188 (2003-08-01), Lee et al.
patent: 2004/0092569 (2004-05-01), Demaine et al.
patent: 2004/0152690 (2004-08-01), Balan et al.
patent: 2004/0248983 (2004-12-01), Morie et al.
patent: 2006/0205802 (2006-09-01), Liu et al.
patent: 2006/0287377 (2006-12-01), Besidski
patent: 2007/0066586 (2007-03-01), Tokumasu et al.
patent: 2008/0015222 (2008-01-01), Besidski et al.
patent: 2300521 (1973-07-01), None
patent: 0149200 (1984-12-01), None
patent: 0419210 (1991-03-01), None
patent: 1312601 (2003-05-01), None
patent: 0882718 (2005-08-01), None
patent: 1186504 (1970-04-01), None
patent: 94/22859 (1994-10-01), None
patent: 99/00115 (1999-01-01), None
patent: 01/12189 (2001-02-01), None
patent: 01/85722 (2001-11-01), None
patent: 01/96336 (2001-12-01), None
patent: 0250031 (2002-06-01), None
patent: 02/072536 (2002-09-01), None
patent: 02/085866 (2002-10-01), None
patent: 02/090326 (2002-11-01), None
patent: 02/100819 (2002-12-01), None
patent: 02/100822 (2002-12-01), None
patent: 03/014064 (2003-02-01), None
patent: 03/022809 (2003-03-01), None
patent: 03/027076 (2003-04-01), None
patent: 03/049702 (2003-06-01), None
patent: 03/053945 (2003-07-01), None
patent: 03/068749 (2003-08-01), None
patent: 2004/000828 (2003-12-01), None
patent: 2004/024154 (2004-03-01), None
patent: 2004/024710 (2004-03-01), None
patent: 2004100865 (2004-11-01), None
patent: 2004/108712 (2004-12-01), None
patent: 2005/021539 (2005-03-01), None
patent: 2005/095327 (2005-12-01), None
patent: 2006033620 (2006-03-01), None
patent: 2007073303 (2007-06-01), None
Caterina, et al., “The capsaicin receptor: a heat-activated ion channel in the pain pathway.” Nature (1997) v. 389, p. 816-824.
Hwang, et al., “Hot channels in airways: pharmacoloty of the vanilloid receptor”. Curr Opin Pharmacol (2002), June, 2 (3), p. 235-242.
Rashid, et al., “Novel Expression of Vanilloid Receptor 1 on Capsaicin-Insensitive Fibers Accounts for the Analgesic Effect of Capsaicin Cream in Neuropathic Pain.” J. Pharmacol Exp Ther. Mar. 2003 304(3), p. 940-948.
Szallasi, A., “Vanilloid (Capsaicin) Receptors in Health and Disease”. Am J. Clin Pathol (2002) 118, p. 110-121.
Tominaga, et al., “The cloned capsaicin receptor integrates multiple pain-producing stimuli.” Neuron (1998) v. 21, p. 531-543.
Walker, K. M., et al., “The VR1 antagonist capsazepine reverses mechanical hyperalgesia in models of inflammatory and neuropathic pain.” J. Pharmacol Exp Ther. Jan. 2003 304(1), p. 56-62.
Yiangou, et al., “Capsaicin receptor VR1 and ATP-gated ion channel P2X3 in human urinary bladder.” BJU Intl (2001), June 87(9), p. 774-779.
Non-final Office Action mailed on Jan. 7, 2008, for U.S. Appl. No. 10/556,229, AstraZeneca ref. No. 101062-1P US.
Non-final Office Action dated Jul. 16, 2007, for U.S. Appl. No. 10/556,229, AstraZeneca ref. No. 101062-1P US.
Gallard, et at., Journal of Enzyme Inhibition and Medicinal Chemistry, vol. 18, No. 2 . 2003, “New N-Pyridinyl (methyl)-N1-Substituted . . . Systemic anti-Inflammatory Agents”, pp. 201-208.
T.L. Gilchrist, “Heterocyclic Chemistry”, 2nd Edition, Longman Scientific andTechnical (1992), pp. 248-282.
Non-final Office Action mailed on May 16, 2008, for U.S. Appl. No. 10/557,806, AstraZeneca reference No. 101101-1P US.
Co-pending U.S. Publication No. 2006-0287377, published on Dec. 21, 2006.
Co-pending U.S. Appl. No. 11/614,346, filed on Dec. 21, 2006.
Co-pending U.S. Publication No. 2008-0015222, published on Jan. 17, 2008.
Co-pending U.S. Publication No. 2006-0205802, published on Sep. 14, 2006.
Non-Final Office Action mailed on Jul. 23, 2008 for U.S. Appl. No. 10/557,806, AstraZeneca reference No. 101101-1P US.
Beilstein Institute for Organic Chemistry, Frankfurt-Main, Germany; XP002291482, BRN 838602 abstract and Kamel et al, J. Prakt. Chem., vol. 31, 1966, pp. 100-105.
Beilstein Institute for Organic Chemistry, Frankfurt-Main, Germany; XP002291483 BRN 926470 abstract and Osman: Kolor. ERT., vol. 11, 1969, p. 118.
Beilstein Institute for Organic Chemistry, Frankfurt-Main, Germany; XP002291484 BRN 311062 abstract & Pinnow; Wiskott: Chem. Ber., vol. 32, 1899, p. 900.
Beilstein Institute for Organic Chemistry, Frankfurt-Main, Germany; XP002291485 BRN 189489 abstract & Foster: J. Chem. Soc., 1957, pp. 4687-4688.
Beilstein Institute for Organic Chemistry, Frankfurt-Main, Germany; XP002291490 BRN 326965 abstract & V. Walter; Kessler: J. Prak. Chem., vol. 2, No. 74, 1906, p. 198.
Kumar et al., “Cyanoethylation of Benzimidazoles: Synthesis & Biological Activities of Some New1-(beta-Cyanoethyl) benzimidazoles & Their Derivatives”, Indian Journal of Chemistry, Oct. 1985, vol. 24B, p. 1098-1101.
Lindberg, et al., “Long-Time Persistence of Superantigen-Producing Staphylococcus aureus Strains in the Intestinal Microflora of Healthy Infants”, Pediatric Research 48:741-747 (2000).
McDonnell, et al., 7-Hydroxynaphthalen-l-yt-Urea and -Amide Antagonists of Human Vanilloid Receptor 1′; Bioorganic & Medicinal Chemistry Letters 14 (2004), pp. 531-534.
Musso, et al., “Indanylidenes. 1 . Design and Synthesis of (E)-2-(4,6-Difluoro-1-indanylidene)acetamide, a Potent, Centrally Acting Muscle Relaxant with Antiinflammatory and Analgesic Activity”; J. Med. Client 2003, 46, pp. 399-408.
Patent Abstracts of Japan vol. 2000, No. 07, Sep. 29, 2000 & JP 2000 095767 A (Takeda Chem Ind Ltd), Apr. 4, 2000.
Sasaki, et al., “Prevention of collagen-induced arthritis with the superantigen Staphylococcal enterotoxin B”, Patho-physiology 4:25-31 (1997), only p. 25 provided.
Soos, et al., “Treatment PL/J mice with the superantigen, staphylococcal enterotoxin B, prevents development of experimental allergic encephalomyelitis”, J Neuroimmunology 43:39-44 (1993), only p. 39 provided.
Willitzer, H. et al., “Synthese und antivirale Wirsamkeit von substituierten 5-Ureido- und 5-Thioureidobenzimidazolderivaten” Pharmazie, Veb Verlag Volk und Gesundheit. Berlin, Germany vol. 33, No. 1, Jan. 1978, pp. 30-38, XP002209435 ISSN: 0031-7144 English Abstract is cited as Accession No. 1978:424221.
STN International, File CAPLUS, accession No. 1978:424221, document No. 89:24221, Willitzer et al., “Synthesis and antiviral activity of substituted 5-ureido- and 5-thioureidobenzimidazole derivates”, & Pharmazie (1978), 33(1) 30-8.
STN International File CAPLUS, accesssion No. 1958:50566, document No. 52-50566, Foster, R. “1-Ethyl-2-methyl-5-nitrobenzimidazole” & Journal of the Chem. Society, Abstracts (1957) 4687-8.
STN International , file CHEMCATS, Accession No. 2000:912544, Apr. 24, 2003, CHS 0297096, 1H-Benzimidazole-1-acetamide, N-[3-(trifluoromethyl)phenyl]-CAS Registry No. 294669-15-1.
STN International, file CHEMCATS, Accession No. 2000 :532079, Apr. 23, 2003, BAS 0238979,1H-Benzimidazole-1-acetamide, N-(3-chlorophenyl)-CAS Registry No. 116488-26-7.
STN International, file CHEMCATS, Accession No. 2001:10738, Apr. 24, 2003, NS11937, 1H-Indole-3-butanamide, N-(4-methylphenyl)-CAS Registry No. 313550-48-0.
STN International, file CHEMCATS, Accession No. 2001:1505160, Apr. 29, 2003, AG-690/40696518,1H-Benzimidazole-l-acetamide, N-(2,3-dichlorophenyl)-, CAS Registry No. 332384-60-8.
STN International, file CHEMCATS, Accession No. 2002:2035573, Jul. 9, 2002, ASN 1816063,1H-Benzimidazole-l-acetamide, N-(3-chloro-4-methylphenyl)—CAS Registry No. 332908-87-9.
STN International, file CHEMCATS, Accession No. 2002:2042451, Jul. 9, 2002, ASN 4428244,1H-Benzimidazole-l-acetamide,N-(5-amnino-2-methylp
Brown William
Johnstone Shawn
Labrecque Denis
Astrazeneca AB
Connolly Bove & Lodge & Hutz LLP
Stockton Laura L.
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