Benzamidine derivatives substituted by cyclic amino acid and cyc

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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5462727, 5462774, 546296, 546297, 546307, 544333, A01N 4340, C07D40100, C07D21172, C07D40300

Patent

active

060082348

ABSTRACT:
This invention is directed to benzamidine derivatives substituted by cyclic amino acid and cyclic hydroxy acid derivatives which are useful as anti-coagulants. This invention is also directed to pharmaceutical compositions containing the compounds of the invention, and methods of using the compounds to treat disease-states characterized by thrombotic activity.

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