Benzamidine derivatives substituted by amino acid and hydroxy ac

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Nitrogen containing other than solely as a nitrogen in an...

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564244, 564225, 564237, 5483355, 5483351, 544335, 544242, 514631, 514396, 514256, A61K 31155, C07C25718

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active

061660884

ABSTRACT:
This invention is directed to benzamidine derivatives substituted by amino acid and hydroxy acid derivatives which are useful as anti-coagulants. This invention is also directed to pharmaceutical compositions containing the compounds of the invention, and methods of using the compounds to treat disease-states characterized by thrombotic activity.

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