Basic cleavage products of elaiophylin and elaiophylin derivativ

Details Basic cleavage products of elaiophylin and elaiophylin derivativ Basic cleavage products of elaiophylin and elaiophylin derivativ

1989-09-14

1992-03-17

Ivy, C. Warren

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514256, 514275, 514336, 514352, 514444, 514447, 514460, 544295, 544323, 544336, 544357, 546251, 546255, 546256, 549 60, 549 68, 549343, 549415, A61K 3150, C07D49310

Patent

active

050969056

ABSTRACT:
The invention relates to elaiophylin derivatives of the formulae (I), (I'), (III) and (III') ##STR1## in which the C.dbd.C double bonds in the 2,3 and 4,5 position may also be hydrogenated and in which R.sup.1, R.sup.2, R.sup.3, R.sup.4 and X have the meanings indicated. The invention furthermore relates to a process for the preparation of these elaiophylin derivatives, and the use thereof as pharmaceuticals, in particular as anthelmintic pharmaceuticals.

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