Azolylacylguanidines as β-secretase inhibitors

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C514S427000

Reexamination Certificate

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07488832

ABSTRACT:
The present invention provides an azolylacylquanidine compound of formula IThe present invention also provides methods for the use thereof to inhibit β-secretase (BACE) and treat β-amyloid deposits and neurofibrillary tangles.

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