Azolopyrimidine-based inhibitors of dipeptidyl peptidase IV...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C544S281000, C544S280000, C544S256000, C514S259300, C514S259310

Reexamination Certificate

active

07635699

ABSTRACT:
Compounds are provided having the formula (I)wherein X for each occurrence is N or C-A, and R, Y, A and n are as defined herein, which compounds are dipeptidyl peptidase IV inhibitors and as such are useful in treating diabetes and micro- and macrovascular complications of diabetes, such as retinopathy, neuropathy, and nephropathy.A method for treating diabetes and related diseases employing the above compounds is also provided.

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