Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1991-03-06
1992-11-10
Morris, Patricia L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
5482622, 5482672, 5482674, 5482678, A61K 3141, C07D21908
Patent
active
051623560
ABSTRACT:
Disclosed herein are azole derivatives or the salts thereof which are represented by the general formula (I): ##STR1## wherein X represents a halogen atom, an alkyl group having 1 to 5 carbon atoms, a haloalkyl group, a phenyl group, a cyano group, or a nitro group, Xs being either the same or different from each other; n represents an integer of 1 to 5; A represents a nitrogen atom or CH; and one of R.sub.1 and R.sub.2 represents an alkyl group having 1 to 5 carbon atoms and the other a hydrogen atom or an alkyl group having 1 to 5 carbon atoms, with the proviso that when n is 1 or 2, X does not represent a halogen atom, an alkyl group having 1 to 5 carbon atoms or a phenyl group, and mycocides comprising an effective amount of azole derivative or medically or veterinarily acceptable salt thereof, said azole derivative being represented by the general formula (II): ##STR2## wherein X represents a halogen atom, an alkyl group having 1 to 5 carbon atoms, a haloalkyl group, a phenyl group, a cyano group, or a nitro group, Xs being either the same or different from each other; n represents an integer of 0 to 5; A represents a nitrogen atom or CH; and R.sub.1 and R.sub.2 respectively represent a hydrogen atom or an alkyl group having 1 to 5 carbon atoms, and a diluent or a carrier which is medically or veterinarily acceptable.
REFERENCES:
patent: 4684396 (1987-08-01), Clough et al.
patent: 4863505 (1989-09-01), Kumazawa et al.
patent: 4938792 (1990-09-01), Kumazawa et al.
Siegel et al, "Arylmethylozoles as fungicides, etc." CA 107:96718s (1987).
Arahira Masato
Ikeda Susumu
Kumazawa Satoru
Saishoji Toshihide
Kureha Kagaku Kogyo Kabushiki Kaisha
Morris Patricia L.
LandOfFree
Azole mycocide and method of treating mycosis does not yet have a rating. At this time, there are no reviews or comments for this patent.
If you have personal experience with Azole mycocide and method of treating mycosis, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Azole mycocide and method of treating mycosis will most certainly appreciate the feedback.
Profile ID: LFUS-PAI-O-2293146