Aza cyclohexapeptide compounds

Details Aza cyclohexapeptide compounds Aza cyclohexapeptide compounds

1993-03-16

1995-01-03

Hill, Jr., Robert J.

Chemistry: natural resins or derivatives; peptides or proteins;

Peptides of 3 to 100 amino acid residues

Cyclic peptides

930270, 930DIG548, 930DIG546, C07K 764

Patent

active

053788044

ABSTRACT:
Aza cyclohexapeptide compounds are disclosed with a nitrogen attached to the cyclohexapeptide ring at the 5-carbon of the 4-hydroxyornithine component. Such compounds are represented by the formula: ##STR1## The compounds are disclosed as having antifungal, antiprotozoal and anti-Pneumocystis carinii activity.

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