Avermectin and avemectin monosaccharide derivatives...

Details Avermectin and avemectin monosaccharide derivatives... Avermectin and avemectin monosaccharide derivatives...

2004-01-30

2009-12-15

Richter, Johann R (Department: 1616)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

C514S450000, C514S210010, C514S320000, C514S321000, C514S337000, C504S100000

Reexamination Certificate

active

07632820

ABSTRACT:
Disclosed are compounds of the formulain which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —SO2—; R1is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2is R3-Z-, R3—O-Z-, R4or -Z-N(R6)(R7); Q is O or —N—R5; R3and R4are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6and R7are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.

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