Arylvinylamide derivatives and pharmaceutical use

Details Arylvinylamide derivatives and pharmaceutical use Arylvinylamide derivatives and pharmaceutical use

1990-11-02

1992-06-16

Raymond, Richard L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Ester doai

514307, 514309, 514311, 514312, 514415, 514418, 514419, 514522, 514630, 546141, 546142, 546146, 546147, 546153, 546155, 546175, 548484, 548485, 548486, 548496, 548503, 558414, 560139, 564219, A61K 31165, C07C23322

Patent

active

051225379

ABSTRACT:
The invention relates to new arylvinylamide derivatives of formula ##STR1## wherein Y is a bicyclic ring system chosen from (A), (B), (C), (D), and (E); ##STR2## in which m is zero, 1 or 2; R is hydrogen, a C.sub.1 -C.sub.6 alkyl or C.sub.1 -C.sub.6 alkanoyl group;

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