Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-05-10
2005-05-10
Bernhardt, Emily (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S210020, C514S210200, C514S217050, C514S252130, C514S253010, C514S254010, C514S254080, C540S200000, C540S354000, C540S362000, C540S451000, C540S481000, C540S524000, C540S598000, C544S230000, C544S360000, C544S372000, C544S373000
Reexamination Certificate
active
06890921
ABSTRACT:
This invention relates to a series of arylsubstituted piperazines, of Formula Ipharmaceutical compositions containing them and intermediates used in their manufacture. The compounds of the invention selectively inhibit binding to the α-1a adrenergic receptor, a receptor which has been implicated in benign prostatic hyperplasia. As such the compounds are potentially useful in the treatment of this and other disease.
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Jolliffe Linda
Li Xiaobing
Maryanoff Cynthia
Mulcahy Linda
Murray William
Bernhardt Emily
Donnelly Laura A.
Ortho-McNeil Pharmaceutical , Inc.
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