Arylglycinamide derivatives and preparative processes therefor

Details Arylglycinamide derivatives and preparative processes therefor Arylglycinamide derivatives and preparative processes therefor

1993-07-20

1995-08-08

Ivy, C. Warren

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514319, 514325, 514330, 514331, 514620, 514423, 514428, 546189, 546195, 546203, 546205, 546220, 546233, 546234, 564164, 564165, 564168, C07C23300, C07D21130, A01N 4340

Patent

active

054399190

ABSTRACT:
Arylglycinamide derivatives represented by a general formula (1) ##STR1## (wherein Ar denotes a phenyl group which may have 1 to 3 substituents or naphthyl group which may have 1 to 3 substituents, R.sub.1 and R.sub.4 denote identically or differently hydrogen atoms or lower alkyl groups with 1 to 3 carbon atoms, R.sub.2 denotes a lower alkyl group with 1 to 6 carbon atoms, cycloalkyl group with 3 to 6 carbon atoms, lower alkyl group with 1 to 4 carbon atoms which may have a phenyl group which may have 1 to 3 substituents, norbornyl group, adamantyl group or phenyl group which may have 1 to 3 substituents, R.sub.3 denotes a hydrogen atom or lower alkyl group with 1 to 6 carbon atoms or it may form a ring constituting alkylene together with R.sub.2, R.sub.5 denotes a lower alkyl group with 1 to 6 carbon atoms or cycloalkyl group with 5 or 6 carbon atoms, R.sub.6 denotes a hydrogen atom or lower alkyl group with 1 to 6 carbon atoms or it may form a ring constituting alkylene together with R.sub.5, and m denotes 2 or 3), and their salts, which function as effective therapeutic drugs for the dysurias such as urinary incontinence and pollakiuria, and the preparative processes therefor are presented.

REFERENCES:
patent: 5153226 (1992-10-01), Chucholowski et al.
Chemical Abstracts, vol. 58, No. 8, Apr. 15, 1963, AN-7913a, S. Kawahara "Alpha-(N-Substituted Animoalkyl) Amino-Alpha-Phenylacetamide".
Chemical Abstracts, vol. 58, No. 8, Apr. 15, 1963, AN-7935d, J. Klosa, "Synthesis of Spasmolytically Active Substances. XVI. Synthesis of Alpha-Phenyl-Alpha-(N,N-Dialkylamnoinoalkyl) Acetamides".

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