Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2007-11-06
2007-11-06
Davis, Zinna N. (Department: 1625)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S317000, C544S336000, C546S192000
Reexamination Certificate
active
10506422
ABSTRACT:
An arylamidine derivative represented by a general formula described below or a salt thereof has an excellent antifungal action and high safety, and it is useful as an antifungal agent with good pharmacokinetics and pharmacodynamic propertieswherein X represents an unsubstituted or substituted lower alkylene or alkenylene group; G1represents an oxygen atom, a sulfur atom, or an imino group; G2represents a carbon atom or a nitrogen atom; Rarepresents at least one group selected from the group consisting of a hydrogen atom, a halogen atom, and unsubstituted or substituted alkyl, cycloalkyl and alkoxy groups; R1represents an unprotected or protected or unsubstituted or substituted amidino group; and R2represents a substituted amino or substituted cyclic amino group, or the like.
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Hayashi Kazuya
Hori Kozo
Kunitani Kazuto
Mitsuyama Junichi
Ojima Katsuji
Davis Zinna N.
Toyama Chemical Co., Ltd.
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